Compile Data Set for Download or QSAR
maximum 50k data
Found 37 Enz. Inhib. hit(s) with all data for entry = 50040330
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataKi:  21.6nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  52.4nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392711(CHEMBL2151380)
Affinity DataKi:  251nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392710(CHEMBL2151379)
Affinity DataKi:  385nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392701(CHEMBL2151370)
Affinity DataKi:  504nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392708(CHEMBL2151377)
Affinity DataKi:  689nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392708(CHEMBL2151377)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392709(CHEMBL2151378)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392707(CHEMBL2151376)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392711(CHEMBL2151380)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392699(CHEMBL2151368)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392700(CHEMBL2151369)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50392702(CHEMBL2151371)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392703(CHEMBL2151372)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392704(CHEMBL2151373)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392705(CHEMBL2151374)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392712(CHEMBL2151381)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392710(CHEMBL2151379)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392709(CHEMBL2151378)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392707(CHEMBL2151376)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392706(CHEMBL2151375)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392705(CHEMBL2151374)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392704(CHEMBL2151373)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392703(CHEMBL2151372)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392702(CHEMBL2151371)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392701(CHEMBL2151370)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392699(CHEMBL2151368)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392700(CHEMBL2151369)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392706(CHEMBL2151375)
Affinity DataKi: >3.00E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392712(CHEMBL2151381)
Affinity DataKi:  3.64E+3nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO cell membranes after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392708(CHEMBL2151377)
Affinity DataEC50:  749nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392710(CHEMBL2151379)
Affinity DataEC50:  371nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392711(CHEMBL2151380)
Affinity DataEC50:  191nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataEC50:  89.6nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50180022(5-(4-chloro-3-methyl-phenyl)-1-(4-methyl-benzyl)-1...)
Affinity DataEC50:  2.10nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Avenue De L'Universit£

Curated by ChEMBL
LigandPNGBDBM50392701(CHEMBL2151370)
Affinity DataEC50:  297nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed