Compile Data Set for Download or QSAR
maximum 50k data
Found 86 Enz. Inhib. hit(s) with all data for entry = 50041756
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50132713(Arachidonic acid derivative | CHEMBL113262 | Methy...)
Affinity DataIC50:  0.331nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50059523((6Z,9Z,12Z,15Z)-1,1,1-trifluorohenicosa-6,9,12,15-...)
Affinity DataIC50:  12.3nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414921(CHEMBL570812)
Affinity DataIC50:  20.4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50132713(Arachidonic acid derivative | CHEMBL113262 | Methy...)
Affinity DataIC50:  26.3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM26736(CHEMBL509860 | LY2183240 | N,N-dimethyl-5-[(4-phen...)
Affinity DataIC50:  38.0nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM26736(CHEMBL509860 | LY2183240 | N,N-dimethyl-5-[(4-phen...)
Affinity DataIC50:  55.0nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414921(CHEMBL570812)
Affinity DataIC50:  77.6nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414919(CHEMBL571699)
Affinity DataIC50:  110nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414940(CHEMBL576697)
Affinity DataIC50:  141nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414953(CHEMBL570565)
Affinity DataIC50:  166nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414944(CHEMBL121556 | NSC-402538)
Affinity DataIC50:  219nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414947(CHEMBL576671)
Affinity DataIC50:  269nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414943(CHEMBL573920)
Affinity DataIC50:  316nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414948(CHEMBL121516 | NSC-527035)
Affinity DataIC50:  316nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414937(CHEMBL583524)
Affinity DataIC50:  347nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414938(CHEMBL571274)
Affinity DataIC50:  437nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414946(CHEMBL571273)
Affinity DataIC50:  479nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414942(CHEMBL569626)
Affinity DataIC50:  490nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414939(CHEMBL570340)
Affinity DataIC50:  741nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414952(CHEMBL570804)
Affinity DataIC50:  741nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414950(CHEMBL585179)
Affinity DataIC50:  813nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50361476(CHEMBL583959)
Affinity DataIC50:  912nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM43362(MLS000069752 | N,N-dimethylcarbamodithioic acid (d...)
Affinity DataIC50:  977nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414920(CHEMBL571495)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414920(CHEMBL571495)
Affinity DataIC50:  2.19E+3nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414951(CHEMBL578805 | US11753371, Compound II-2h)
Affinity DataIC50:  4.07E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414940(CHEMBL576697)
Affinity DataIC50:  4.79E+3nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414941(CHEMBL570572)
Affinity DataIC50:  5.01E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50128581(Biphenyl-3-yl-carbamic acid cyclohexyl ester | CHE...)
Affinity DataIC50:  5.75E+3nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414925(CHEMBL571701)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50059523((6Z,9Z,12Z,15Z)-1,1,1-trifluorohenicosa-6,9,12,15-...)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414945(CHEMBL583000)
Affinity DataIC50:  6.92E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414922(CHEMBL570577)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414923(CHEMBL573921)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414936(CHEMBL120082 | NSC-608475 | US11753371, Compound I...)
Affinity DataIC50:  9.55E+3nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50128581(Biphenyl-3-yl-carbamic acid cyclohexyl ester | CHE...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414935(CHEMBL567397)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414924(DITHIODIMORPHOLINE)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414949(CHEMBL571700)
Affinity DataIC50:  1.23E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414926(CHEMBL583322)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase, mitochondrial(Rattus norvegicus)
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414919(CHEMBL571699)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of recombinant rat ALDH activity in liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414927(CHEMBL582931)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414934(CHEMBL570813)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414943(CHEMBL573920)
Affinity DataIC50:  2.51E+4nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414952(CHEMBL570804)
Affinity DataIC50:  3.39E+4nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAldehyde dehydrogenase, mitochondrial(Rattus norvegicus)
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)
Affinity DataIC50:  3.98E+4nMAssay Description:Inhibition of recombinant rat ALDH activity in liver mitochondriaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM43362(MLS000069752 | N,N-dimethylcarbamodithioic acid (d...)
Affinity DataIC50:  4.47E+4nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414944(CHEMBL121556 | NSC-402538)
Affinity DataIC50:  7.94E+4nMAssay Description:Inhibition of human recombinant FAAH-maltose binding proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Universite Catholique De Louvain

Curated by ChEMBL
LigandPNGBDBM50414932(CHEMBL570228)
Affinity DataIC50:  9.55E+4nMAssay Description:Inhibition of human MGL activity using [3H]2-oleoylglycerol substrate by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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