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Found 31 Enz. Inhib. hit(s) with all data for entry = 50043408
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  4.42E+3nMAssay Description:Reversible inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 s...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440686(CHEMBL2430765)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440667(CHEMBL2430662)
Affinity DataIC50:  1.96E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440692(CHEMBL2430667)
Affinity DataIC50:  2.49E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440675(CHEMBL2430654)
Affinity DataIC50:  3.76E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440668(CHEMBL2430661)
Affinity DataIC50:  4.02E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440673(CHEMBL2430656)
Affinity DataIC50:  4.05E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440663(CHEMBL2430666)
Affinity DataIC50:  4.28E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440665(CHEMBL2430664)
Affinity DataIC50:  4.53E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440676(CHEMBL2430653)
Affinity DataIC50:  4.74E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440664(CHEMBL2430665)
Affinity DataIC50:  4.85E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440674(CHEMBL2430655)
Affinity DataIC50:  4.86E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440685(CHEMBL2430766)
Affinity DataIC50:  4.90E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440677(CHEMBL2430652)
Affinity DataIC50:  4.94E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440671(CHEMBL2430658)
Affinity DataIC50:  4.96E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440669(CHEMBL2430660)
Affinity DataIC50:  5.01E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440672(CHEMBL2430657)
Affinity DataIC50:  5.03E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440670(CHEMBL2430659)
Affinity DataIC50:  5.25E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440666(CHEMBL2430663)
Affinity DataIC50:  5.43E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440682(CHEMBL2430769)
Affinity DataIC50:  5.81E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440691(CHEMBL2430668)
Affinity DataIC50:  6.02E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440681(CHEMBL2430770)
Affinity DataIC50:  6.02E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440687(CHEMBL2430764)
Affinity DataIC50:  6.04E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440679(CHEMBL2430651)
Affinity DataIC50:  6.12E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440689(CHEMBL2430670)
Affinity DataIC50:  6.12E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440684(CHEMBL2430767)
Affinity DataIC50:  6.15E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440690(CHEMBL2430669)
Affinity DataIC50:  6.22E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440680(CHEMBL2430650)
Affinity DataIC50:  6.28E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440688(CHEMBL2430671)
Affinity DataIC50:  6.49E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440678(CHEMBL2429876)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))TBA
LigandPNGBDBM50440683(CHEMBL2430768)
Affinity DataIC50:  6.58E+4nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine as substrate incubated for 20 mins prior to substrate addition measured every 30 secs for 4 m...More data for this Ligand-Target Pair
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