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Found 80 Enz. Inhib. hit(s) with all data for entry = 50005619
TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50094696(1-(2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4]triazol...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109473(1-(8-Ethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109455(1-(4-Chloro-phenyl)-3-(8-ethyl-2-furan-2-yl-8H-pyr...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109441(1-(benzo[d][1,3]dioxol-5-yl)-3-(2-(furan-2-yl)-8-m...)
Affinity DataKi:  0.240nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109475(1-(benzo[d][1,3]dioxol-5-yl)-3-(8-ethyl-2-(furan-2...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109462(1-(4-Fluoro-phenyl)-3-(2-furan-2-yl-8-propyl-8H-py...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109454(1-(4-Chloro-phenyl)-3-(2-furan-2-yl-8-methyl-8H-py...)
Affinity DataKi:  0.290nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109480(1-(2-Chloro-phenyl)-3-(8-ethyl-2-furan-2-yl-8H-pyr...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109446(1-(benzo[d][1,3]dioxol-5-yl)-3-(2-(furan-2-yl)-8-p...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50094687(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.320nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109434(1-(4-Fluoro-phenyl)-3-(2-furan-2-yl-8-methyl-8H-py...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109458(1-(4-Chloro-phenyl)-3-(2-furan-2-yl-8-propyl-8H-py...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109489(1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109437(1-(4-Bromo-phenyl)-3-(8-ethyl-2-furan-2-yl-8H-pyra...)
Affinity DataKi:  0.370nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109469(1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109463(1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109439(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109451(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.430nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109435(1-(4-Bromo-phenyl)-3-(2-furan-2-yl-8-propyl-8H-pyr...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109477(1-(4-Bromo-phenyl)-3-(2-furan-2-yl-8-methyl-8H-pyr...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50085371(1-(8-Allyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.480nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109484(1-(benzo[d][1,3]dioxol-5-yl)-3-(8-butyl-2-(furan-2...)
Affinity DataKi:  0.500nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50094683(1-(3-Chloro-phenyl)-3-(2-furan-2-yl-8H-pyrazolo[4,...)
Affinity DataKi:  0.500nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109479(1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.511nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109467(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.550nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109452(1-(8-Ethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.560nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109470(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50082418(1-(8-ethyl-2-(furan-2-yl)-8H-pyrazolo[4,3-e][1,2,4...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109436(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50094699(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109471(1-(8-Ethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.650nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109487(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109460(1-(2-Chloro-phenyl)-3-(2-furan-2-yl-8-propyl-8H-py...)
Affinity DataKi:  0.710nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109457(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.719nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109468(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.740nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109464(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109474(1-(2-(furan-2-yl)-8-methyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50094686(1-(8-tert-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM85618(CHEMBL302765 | J1.251.181G | MRE 3008F20)
Affinity DataKi:  0.800nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109448(1-(2-(furan-2-yl)-8-propyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  0.809nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109453(CHEMBL341376 | N-(2-(furan-2-yl)-8-methyl-8H-pyraz...)
Affinity DataKi:  0.809nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109447(1-(8-Ethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.859nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109466(1-(8-Ethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.859nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109440(1-(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.859nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM85619(1-(3-chlorophenyl)-3-[2-(furan-2-yl)-8-propyl-8H-p...)
Affinity DataKi:  0.910nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109476(1-(4-Bromo-phenyl)-3-(8-butyl-2-furan-2-yl-8H-pyra...)
Affinity DataKi:  0.910nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109459(1-(2-Chloro-phenyl)-3-(2-furan-2-yl-8-methyl-8H-py...)
Affinity DataKi:  0.910nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109444(1-(8-Ethyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]t...)
Affinity DataKi:  0.971nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50109482(CHEMBL165073 | N-(8-Ethyl-2-furan-2-yl-8H-pyrazolo...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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TargetAdenosine receptor A3(Homo sapiens (Human))TBA
LigandPNGBDBM50158777(1-Cyclohexyl-3-(2-furan-2-yl-8-methyl-8H-pyrazolo[...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
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