Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 208
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228095(US9556160, ex 556)
Affinity DataIC50:  2.70nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228072(US9556160, ex 63)
Affinity DataIC50:  3.40nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228098(US9556160, ex 559 | US9556160, ex 567)
Affinity DataIC50:  4.30nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228098(US9556160, ex 559 | US9556160, ex 567)
Affinity DataIC50:  4.30nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228069(US9556160, ex 11)
Affinity DataIC50:  5.20nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228073(US9556160, ex 74)
Affinity DataIC50:  5.30nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228105(US9556160, ex 566)
Affinity DataIC50:  6.30nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228070(US9556160, ex 29)
Affinity DataIC50:  7.20nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228099(US9556160, ex 560)
Affinity DataIC50:  9nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228100(US9556160, ex 561)
Affinity DataIC50:  9.60nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228074(US9556160, ex 81)
Affinity DataIC50:  9.70nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228096(US9556160, ex 557)
Affinity DataIC50:  11nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228089(US9556160, ex 335)
Affinity DataIC50:  11nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228087(US9556160, ex 316)
Affinity DataIC50:  11nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228101(US9556160, ex 562)
Affinity DataIC50:  14nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228076(US9556160, ex 105)
Affinity DataIC50:  14nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228090(US9556160, ex 551)
Affinity DataIC50:  14nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228079(US9556160, ex 126)
Affinity DataIC50:  15nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228104(US9556160, ex 565)
Affinity DataIC50:  19nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228103(US9556160, ex 564)
Affinity DataIC50:  19nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228085(US9556160, ex 300)
Affinity DataIC50:  19nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228084(US9556160, ex 293)
Affinity DataIC50:  19nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228083(US9556160, ex 273)
Affinity DataIC50:  19nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228092(US9556160, ex 553)
Affinity DataIC50:  20nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228102(US9556160, ex 563)
Affinity DataIC50:  20nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228094(US9556160, ex 555)
Affinity DataIC50:  20nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228093(US9556160, ex 554)
Affinity DataIC50:  21nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228071(US9556160, ex 52)
Affinity DataIC50:  23nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228097(US9556160, ex 558)
Affinity DataIC50:  23nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228075(US9556160, ex 83)
Affinity DataIC50:  25nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228082(US9556160, ex 220)
Affinity DataIC50:  25nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228091(US9556160, ex 552)
Affinity DataIC50:  25nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228078(US9556160, ex 118)
Affinity DataIC50:  29nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228077(US9556160, ex 110)
Affinity DataIC50:  32nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228081(US9556160, ex 178)
Affinity DataIC50:  33nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228086(US9556160, ex 304)
Affinity DataIC50:  34nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228080(US9556160, ex 157)
Affinity DataIC50:  49nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Astellas Pharma

US Patent
LigandPNGBDBM228088(US9556160, ex 322)
Affinity DataIC50:  51nMT: 2°CAssay Description:A human VAP-1 enzyme (SSAO) (reference: J Exp Med. 1998 Jul. 6; 188(1): 17 to 27) activity was measured by a radiochemistry-enzymatic assay using 14C...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent