Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 3307
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31183(thiazol-2-amine, 14)
Affinity DataIC50:  700nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31183(thiazol-2-amine, 14)
Affinity DataIC50:  1.10E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31175(thiazol-2-amine, 5)
Affinity DataIC50:  3.00E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31186(thiazol-2-amine, 18)
Affinity DataIC50:  3.20E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31185(thiazol-2-amine, 17)
Affinity DataIC50:  3.20E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31182(thiazol-2-amine, 13)
Affinity DataIC50:  3.30E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31185(thiazol-2-amine, 17)
Affinity DataIC50:  3.50E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31182(thiazol-2-amine, 13)
Affinity DataIC50:  5.00E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31178(thiazol-2-amine, 8)
Affinity DataIC50:  6.50E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31179(thiazol-2-amine, 9)
Affinity DataIC50:  6.50E+3nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31175(thiazol-2-amine, 5)
Affinity DataIC50:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31178(thiazol-2-amine, 8)
Affinity DataIC50:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31179(thiazol-2-amine, 9)
Affinity DataIC50:  1.20E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31176(thiazol-2-amine, 6)
Affinity DataIC50:  1.20E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31187(thiazol-2-amine, 19)
Affinity DataIC50:  1.65E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31188(thiazol-2-amine, 20)
Affinity DataIC50:  1.70E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31177(thiazol-2-amine, 7)
Affinity DataIC50:  1.80E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31188(thiazol-2-amine, 20)
Affinity DataIC50:  1.80E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31176(thiazol-2-amine, 6)
Affinity DataIC50:  1.85E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31184(thiazol-2-amine, 16)
Affinity DataIC50:  2.05E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31181(thiazol-2-amine, 11)
Affinity DataIC50:  2.25E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31186(thiazol-2-amine, 18)
Affinity DataIC50:  2.35E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31180(thiazol-2-amine, 10)
Affinity DataIC50:  3.60E+4nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31177(thiazol-2-amine, 7)
Affinity DataIC50:  4.05E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31184(thiazol-2-amine, 16)
Affinity DataIC50:  4.90E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31181(thiazol-2-amine, 11)
Affinity DataIC50:  6.10E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31187(thiazol-2-amine, 19)
Affinity DataIC50:  6.60E+4nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31180(thiazol-2-amine, 10)
Affinity DataIC50:  1.10E+5nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31189(thiazol-2-amine, 21)
Affinity DataIC50: >5.00E+5nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31189(thiazol-2-amine, 21)
Affinity DataIC50: >5.00E+5nMpH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31194(thiazol-2-amine, 12)
Affinity DataIC50: >7.00E+5nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31195(thiazol-2-amine, 15)
Affinity DataIC50: >1.00E+6nMAssay Description:His6-CBFbeta (1-141) was expressed and purified with the exception of the protease cleavage step. Cerulean-Runt domain fusion protein (Runx1 41-190) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31190(thiazol-2-amine, 1)
Affinity DatapH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31191(thiazol-2-amine, 2)
Affinity DatapH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31192(thiazol-2-amine, 3)
Affinity DatapH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31195(thiazol-2-amine, 15)
Affinity DatapH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31194(thiazol-2-amine, 12)
Affinity DatapH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRunt-related transcription factor 1(Homo sapiens (Human))
University Of Virginia At Charlottesville

LigandPNGBDBM31193(thiazol-2-amine, 4)
Affinity DatapH: 7.5 T: 2°CAssay Description:For the FRET measurements, the Cerulean-Runt (Runx1 41-190) and Venus-CBFbeta (1-141) fusion proteins were dialyzed into FRET assay buffer. Protein c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed