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Found 25 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50041822
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416337(CHEMBL1173725)
Affinity DataEC50:  955nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416336(CHEMBL380346)
Affinity DataEC50:  135nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416339(CHEMBL1173081)
Affinity DataEC50:  724nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416340(CHEMBL1173106)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416341(CHEMBL1173170)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416342(CHEMBL1172763)
Affinity DataEC50:  676nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416343(CHEMBL1172764)
Affinity DataEC50:  2.95E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416344(CHEMBL1172605)
Affinity DataEC50:  933nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416345(CHEMBL1172234)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416346(CHEMBL1173147)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416347(CHEMBL1173399)
Affinity DataEC50:  148nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416348(CHEMBL1173400)
Affinity DataEC50:  2.88E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416349(CHEMBL1173171)
Affinity DataEC50:  5.25E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416350(CHEMBL1171808)
Affinity DataEC50:  51.3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416351(CHEMBL1173172)
Affinity DataEC50:  501nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416352(CHEMBL1173492)
Affinity DataEC50:  692nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416353(CHEMBL1172223)
Affinity DataEC50:  263nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416354(CHEMBL1172224)
Affinity DataEC50:  2.29E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416355(CHEMBL1172407)
Affinity DataEC50:  1.17E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416356(CHEMBL1172180)
Affinity DataEC50:  2.24E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50164424(3-(4-Chloro-phenyl)-3-(2-dimethylamino-ethyl)-isoc...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416357(CHEMBL1170888)
Affinity DataEC50:  4.17E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416358(CHEMBL1173239)
Affinity DataEC50:  1.95E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416359(CHEMBL1173689)
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2(Homo sapiens (Human))
University Of Gothenburg

Curated by ChEMBL
LigandPNGBDBM50416338(CHEMBL1172604)
Affinity DataEC50:  1.74E+3nMAssay Description:Agonist activity against human urotensin 2 receptor expressed in human NIH373 cells assessed as beta-galactosidase activity after 5 days by R-SAT ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed