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Found 38 Enz. Inhib. hit(s) with all data for assayid = 1 entry = 50047523
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173112(CHEMBL3810110)
Affinity DataIC50:  0.300nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173116(CHEMBL3810145)
Affinity DataIC50:  1.30nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173101(CHEMBL3808572)
Affinity DataIC50:  1.90nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173108(CHEMBL3809490)
Affinity DataIC50:  1.90nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50160154(1-(3-Hydroxy-propyl)-5-((R)-2-{2-[2-(2,2,2-trifluo...)
Affinity DataIC50:  1.90nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172992(CHEMBL3809248)
Affinity DataIC50:  1.90nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173115(CHEMBL3809840)
Affinity DataIC50:  2.20nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172997(CHEMBL3808726)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172994(CHEMBL3810346)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173110(CHEMBL3808511)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173109(CHEMBL3809093)
Affinity DataIC50:  2.70nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172998(CHEMBL3809175)
Affinity DataIC50:  2.90nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173004(CHEMBL3808896)
Affinity DataIC50:  2.90nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173003(CHEMBL3187195)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173114(CHEMBL3810005)
Affinity DataIC50:  3.20nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173100(CHEMBL3809794)
Affinity DataIC50:  3.70nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173113(CHEMBL3809630)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173117(CHEMBL3809319)
Affinity DataIC50:  4.40nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173005(CHEMBL3809600)
Affinity DataIC50:  4.60nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173002(CHEMBL3808408)
Affinity DataIC50:  4.80nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173111(CHEMBL3810220)
Affinity DataIC50:  7.60nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173104(CHEMBL3809676)
Affinity DataIC50:  8nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173006(CHEMBL3808417)
Affinity DataIC50:  8.10nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172999(CHEMBL3808632)
Affinity DataIC50:  8.60nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173000(CHEMBL3808878)
Affinity DataIC50:  14nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173105(CHEMBL3810401)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172996(CHEMBL3808717)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173118(CHEMBL3808999)
Affinity DataIC50:  21nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173103(CHEMBL3809532)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173001(CHEMBL3810198)
Affinity DataIC50:  26nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172991(CHEMBL3809781)
Affinity DataIC50:  28nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172993(CHEMBL3810187)
Affinity DataIC50:  38nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173102(CHEMBL3809032)
Affinity DataIC50:  57nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173107(CHEMBL3809500)
Affinity DataIC50:  58nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172995(CHEMBL3808981)
Affinity DataIC50:  63nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50172990(CHEMBL3808595)
Affinity DataIC50:  71nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173106(CHEMBL3809543)
Affinity DataIC50:  324nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Chengdu University

Curated by ChEMBL
LigandPNGBDBM50173099(CHEMBL3809314)
Affinity DataIC50:  454nMAssay Description:Antagonist activity at human alpha-1A adrenergic receptor transfected in HEK293 cells assessed as reduction in agonist-induced calcium mobilization a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed