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Compile Data Set for Download or QSAR

Found 22 hits Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50046221   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100615
PNG
(E-7050 | E7050 | GOLVATINIB | Golvatinib)
Show SMILES CN1CCN(CC1)C1CCN(CC1)C(=O)Nc1cc(Oc2ccc(NC(=O)C3(CC3)C(=O)Nc3ccc(F)cc3)c(F)c2)ccn1
Show InChI InChI=1S/C33H37F2N7O4/c1-40-16-18-41(19-17-40)24-9-14-42(15-10-24)32(45)39-29-21-26(8-13-36-29)46-25-6-7-28(27(35)20-25)38-31(44)33(11-12-33)30(43)37-23-4-2-22(34)3-5-23/h2-8,13,20-21,24H,9-12,14-19H2,1H3,(H,37,43)(H,38,44)(H,36,39,45)
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Article
PubMed
n/an/a 20n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100627
PNG
(CHEMBL3321901)
Show SMILES Fc1ccc(cc1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H14FN5/c22-14-7-5-13(6-8-14)20-26-18-10-9-15(11-19(18)27-20)25-21-16-3-1-2-4-17(16)23-12-24-21/h1-12H,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 50n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100624
PNG
(CHEMBL3321904)
Show SMILES Clc1ccc(cc1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H14ClN5/c22-14-7-5-13(6-8-14)20-26-18-10-9-15(11-19(18)27-20)25-21-16-3-1-2-4-17(16)23-12-24-21/h1-12H,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 150n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100623
PNG
(CHEMBL3321905)
Show SMILES Brc1ccc(cc1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H14BrN5/c22-14-7-5-13(6-8-14)20-26-18-10-9-15(11-19(18)27-20)25-21-16-3-1-2-4-17(16)23-12-24-21/h1-12H,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 560n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100614
PNG
(CHEMBL3321892)
Show SMILES N(c1ccc2nc([nH]c2c1)-c1ccccc1)c1ncnc2ccccc12
Show InChI InChI=1S/C21H15N5/c1-2-6-14(7-3-1)20-25-18-11-10-15(12-19(18)26-20)24-21-16-8-4-5-9-17(16)22-13-23-21/h1-13H,(H,25,26)(H,22,23,24)
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PubMed
n/an/a 1.34E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100628
PNG
(CHEMBL3321900)
Show SMILES Fc1cccc(c1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H14FN5/c22-14-5-3-4-13(10-14)20-26-18-9-8-15(11-19(18)27-20)25-21-16-6-1-2-7-17(16)23-12-24-21/h1-12H,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 1.50E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100618
PNG
(CHEMBL3321910)
Show SMILES Clc1ccc(cc1Cl)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H13Cl2N5/c22-15-7-5-12(9-16(15)23)20-27-18-8-6-13(10-19(18)28-20)26-21-14-3-1-2-4-17(14)24-11-25-21/h1-11H,(H,27,28)(H,24,25,26)
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PubMed
n/an/a 1.53E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100617
PNG
(CHEMBL3321911)
Show SMILES Clc1cc(Cl)cc(c1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H13Cl2N5/c22-13-7-12(8-14(23)9-13)20-27-18-6-5-15(10-19(18)28-20)26-21-16-3-1-2-4-17(16)24-11-25-21/h1-11H,(H,27,28)(H,24,25,26)
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PubMed
n/an/a 3.58E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100625
PNG
(CHEMBL3321903)
Show SMILES Clc1cccc(c1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H14ClN5/c22-14-5-3-4-13(10-14)20-26-18-9-8-15(11-19(18)27-20)25-21-16-6-1-2-7-17(16)23-12-24-21/h1-12H,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 4.24E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100633
PNG
(CHEMBL3321895)
Show SMILES Cc1ccc(cc1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C22H17N5/c1-14-6-8-15(9-7-14)21-26-19-11-10-16(12-20(19)27-21)25-22-17-4-2-3-5-18(17)23-13-24-22/h2-13H,1H3,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 4.54E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100630
PNG
(CHEMBL3321898)
Show SMILES CCc1ccc(cc1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C23H19N5/c1-2-15-7-9-16(10-8-15)22-27-20-12-11-17(13-21(20)28-22)26-23-18-5-3-4-6-19(18)24-14-25-23/h3-14H,2H2,1H3,(H,27,28)(H,24,25,26)
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PubMed
n/an/a 7.30E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100629
PNG
(CHEMBL3321899)
Show SMILES Fc1ccccc1-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H14FN5/c22-16-7-3-1-5-14(16)21-26-18-10-9-13(11-19(18)27-21)25-20-15-6-2-4-8-17(15)23-12-24-20/h1-12H,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 7.48E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100616
PNG
(CHEMBL3321912)
Show SMILES Fc1ccc(Br)c(c1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H13BrFN5/c22-16-7-5-12(23)9-15(16)21-27-18-8-6-13(10-19(18)28-21)26-20-14-3-1-2-4-17(14)24-11-25-20/h1-11H,(H,27,28)(H,24,25,26)
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PubMed
n/an/a 7.85E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100612
PNG
(CHEMBL3321894)
Show SMILES Cc1cccc(c1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C22H17N5/c1-14-5-4-6-15(11-14)21-26-19-10-9-16(12-20(19)27-21)25-22-17-7-2-3-8-18(17)23-13-24-22/h2-13H,1H3,(H,26,27)(H,23,24,25)
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PubMed
n/an/a 8.80E+3n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100621
PNG
(CHEMBL3321907)
Show SMILES FC(F)(F)c1cccc(c1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C22H14F3N5/c23-22(24,25)14-5-3-4-13(10-14)20-29-18-9-8-15(11-19(18)30-20)28-21-16-6-1-2-7-17(16)26-12-27-21/h1-12H,(H,29,30)(H,26,27,28)
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PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100620
PNG
(CHEMBL3321908)
Show SMILES FC(F)(F)c1ccc(cc1)-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C22H14F3N5/c23-22(24,25)14-7-5-13(6-8-14)20-29-18-10-9-15(11-19(18)30-20)28-21-16-3-1-2-4-17(16)26-12-27-21/h1-12H,(H,29,30)(H,26,27,28)
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PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100631
PNG
(CHEMBL3321897)
Show SMILES Oc1ccccc1-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H15N5O/c27-19-8-4-2-6-15(19)21-25-17-10-9-13(11-18(17)26-21)24-20-14-5-1-3-7-16(14)22-12-23-20/h1-12,27H,(H,25,26)(H,22,23,24)
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PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100626
PNG
(CHEMBL3321902)
Show SMILES Clc1ccccc1-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H14ClN5/c22-16-7-3-1-5-14(16)21-26-18-10-9-13(11-19(18)27-21)25-20-15-6-2-4-8-17(15)23-12-24-20/h1-12H,(H,26,27)(H,23,24,25)
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PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100619
PNG
(CHEMBL3321909)
Show SMILES Clc1cccc(Cl)c1-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C21H13Cl2N5/c22-14-5-3-6-15(23)19(14)21-27-17-9-8-12(10-18(17)28-21)26-20-13-4-1-2-7-16(13)24-11-25-20/h1-11H,(H,27,28)(H,24,25,26)
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PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100613
PNG
(CHEMBL3321893)
Show SMILES Cc1ccccc1-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C22H17N5/c1-14-6-2-3-7-16(14)22-26-19-11-10-15(12-20(19)27-22)25-21-17-8-4-5-9-18(17)23-13-24-21/h2-13H,1H3,(H,26,27)(H,23,24,25)
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PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100622
PNG
(CHEMBL3321906)
Show SMILES FC(F)(F)c1ccccc1-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C22H14F3N5/c23-22(24,25)16-7-3-1-5-14(16)21-29-18-10-9-13(11-19(18)30-21)28-20-15-6-2-4-8-17(15)26-12-27-20/h1-12H,(H,29,30)(H,26,27,28)
PDB
MMDB

KEGG

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DrugBank
antibodypedia
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PC cid
PC sid
UniChem

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Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair
Hepatocyte growth factor receptor


(Homo sapiens (Human))
BDBM50100632
PNG
(CHEMBL3321896)
Show SMILES COc1ccccc1-c1nc2ccc(Nc3ncnc4ccccc34)cc2[nH]1
Show InChI InChI=1S/C22H17N5O/c1-28-20-9-5-3-7-16(20)22-26-18-11-10-14(12-19(18)27-22)25-21-15-6-2-4-8-17(15)23-13-24-21/h2-13H,1H3,(H,26,27)(H,23,24,25)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
PC cid
PC sid
UniChem

Similars

AffyNet 
Article
PubMed
n/an/a>1.00E+4n/an/an/an/an/an/a



Jiangsu Key Laboratory of Drug Design and Optimization, Department of Medicinal Chemistry, China Pharmaceutical University, Nanjing 210009, PR China. Electronic address: shilei@cpu.edu.cn.

Curated by ChEMBL


Assay Description
Inhibition of human recombinant c-Met pre-incubated for 5 mins before ATP/substrate peptide cocktail addition measured after 30 mins by colorimetric ...


Bioorg Med Chem 22: 4735-44 (2014)

More data for this
Ligand-Target Pair