Compile Data Set for Download or QSAR
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Found 6 of ph data with Target = 'Trans-sialidase'
TargetTrans-sialidase(Trypanosoma cruzi)
University Of British Columbia

LigandPNGBDBM84698(Quinolinone derivative, 9)
Affinity DataKi:  400nM ΔG°:  -37.7kJ/mole IC50:  600nMpH: 7.6 T: 2°CAssay Description:Inhibition assay using trans-sialidase, a membrane-associated protein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrans-sialidase(Trypanosoma cruzi)
University Of British Columbia

LigandPNGBDBM50174833(CHEMBL199442 | N-(3-(3-(3,4-dihydroxyphenyl)acrylo...)
Affinity DataKi:  3.70E+3nM ΔG°:  -32.0kJ/mole IC50:  2.50E+3nMpH: 7.6 T: 2°CAssay Description:Inhibition assay using trans-sialidase, a membrane-associated protein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrans-sialidase(Trypanosoma cruzi)
University Of British Columbia

LigandPNGBDBM50174837(4'-(p-toluenesulfonamide)-3,4-dihydroxy chalcone |...)
Affinity DataKi:  4.60E+3nM ΔG°:  -31.5kJ/mole IC50:  900nMpH: 7.6 T: 2°CAssay Description:Inhibition assay using trans-sialidase, a membrane-associated protein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrans-sialidase(Trypanosoma cruzi)
University Of British Columbia

LigandPNGBDBM84697(Quinolinone derivative, 8)
Affinity DataIC50:  3.00E+4nMpH: 7.6 T: 2°CAssay Description:Inhibition assay using trans-sialidase, a membrane-associated protein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrans-sialidase(Trypanosoma cruzi)
University Of British Columbia

LigandPNGBDBM50174835(4'-(4-toluenesulfonamido)-4-hydroxychalcone | 4'-(...)
Affinity DataIC50:  7.30E+4nMpH: 7.6 T: 2°CAssay Description:Inhibition assay using trans-sialidase, a membrane-associated protein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrans-sialidase(Trypanosoma cruzi)
University Of British Columbia

LigandPNGBDBM50174834(CHEMBL382280 | N-(3-(3-(4-hydroxyphenyl)acryloyl)p...)
Affinity DataIC50:  3.70E+4nMpH: 7.6 T: 2°CAssay Description:Inhibition assay using trans-sialidase, a membrane-associated protein.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed