Affinity DataEC50: 0.0490nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.0575nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at wild type human NK1 receptor expressed in HEK293 cells assessed as increase in [3H]IP accumulation after 20 minsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 0.600nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Compound was evaluated for effective dose against Muscular receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Compound was evaluated for effective dose against muscular receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Compound was evaluated for effective dose against Neuronal receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 6.90nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 13.5nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 24.4nMAssay Description:Displacement of [3H]SR140333 from human recombinant NK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 38nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Effective dose of the compound was measured on NK1 receptors of guinea pig ileum for maximal contraction in the presence of 3*10e-7 M atropineMore data for this Ligand-Target Pair
Affinity DataEC50: 44nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 60nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 61nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 63nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 68nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 86nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: >100nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 160nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Tested for the biological activity and selectivity against NK-1 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 188nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 307nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Effective concentration to activate Tachykinin receptor 1 in guinea pig ileum(GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 545nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair