Compile Data Set for Download or QSAR
maximum 50k data
Found 112 of ec50 data for polymerid = 50001092,50002004,50004899,50002004
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50332462(2-(2-methyl-4-((4-methyl-2-(4-(trifluoromethyl)phe...)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at mouse PPAR-delta expressed in african green monkey CV-1 cells after 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312479(2-(4-((4-(6-Morpholinopyridin-3-yl)-5-(4-(trifluor...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615952(CHEMBL5267473)
Affinity DataEC50:  5.80nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615955(CHEMBL5283926)
Affinity DataEC50:  6.10nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615962(CHEMBL5272996)
Affinity DataEC50:  6.20nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615954(CHEMBL5290870)
Affinity DataEC50:  6.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615966(CHEMBL5289740)
Affinity DataEC50:  6.90nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312476(CHEMBL1080699 | {4-[4-(6-Isopropoxypyridin-3-yl)-5...)
Affinity DataEC50:  7nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615964(CHEMBL5277165)
Affinity DataEC50:  7.5nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50539514(CHEMBL4649683)
Affinity DataEC50:  7.90nMAssay Description:Modulator activity at mouse PPARdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312422(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312421(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-(trifluorometho...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312478(2-(4-((4-(2-Isopropoxypyrimidin-5-yl)-5-(4-(triflu...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615947(CHEMBL5278892)
Affinity DataEC50:  12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615963(CHEMBL5290260)
Affinity DataEC50:  12nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312475(2-(4-((4-(6-Isopropoxypyridin-3-yl)-5-(4-(trifluor...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312469(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-propylphenyl)th...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50106105(2-[3-(3-{(2,4-Bis-trifluoromethyl-benzyl)-[2-(4-tr...)
Affinity DataEC50:  19nMAssay Description:Agonist activity against PPAR deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50584465(CHEMBL5084377)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta in Cos7 cells transfected with pBIND and pGL4.35 Gal4 UAS Luc reporter plasmid by measuring luciferase activity i...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  20nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312467(2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-isopropo...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50085040(CHEMBL278994 | L-796449 | {3-Chloro-4-[3-(3-phenyl...)
Affinity DataEC50:  23nMAssay Description:Agonist activity for murine PPAR delta receptor in transcriptional activation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615960(CHEMBL5289017)
Affinity DataEC50:  24nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615946(CHEMBL5271479)
Affinity DataEC50:  25nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615961(CHEMBL5268424)
Affinity DataEC50:  26nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312424(CHEMBL1080349 | {4-[4-(4-Isopropoxyphenyl)-5-(4-tr...)
Affinity DataEC50:  26nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615951(CHEMBL5285352)
Affinity DataEC50:  27nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615958(CHEMBL5279586)
Affinity DataEC50:  28nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312470(2-(4-((4-(4-Isopropoxyphenyl)-5-(4-biphenyl)thiazo...)
Affinity DataEC50:  29nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312477(2-(4-((4-(2-Methoxypyrimidin-5-yl)-5-(4-propylphen...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataEC50:  30nMAssay Description:Activity against murine PPAR delta receptorMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312472(2-(4-((5-(4-Biphenyl)-4-(pyridin-3-yl)oxazol-2-yl)...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312425(2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluor...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615957(CHEMBL5268646)
Affinity DataEC50:  34nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615959(CHEMBL5273427)
Affinity DataEC50:  39nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312468(2-(4-((4-(4-Isopropoxyphenyl)-5-(3-(trifluorometho...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615950(CHEMBL5288454)
Affinity DataEC50:  46nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615948(CHEMBL5281528)
Affinity DataEC50:  47nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615949(CHEMBL5278648)
Affinity DataEC50:  47nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596502(CHEMBL5180328)
Affinity DataEC50:  49nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  54nMAssay Description:Agonist activity at mouse PPAR delta expressed in HEK293 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615953(CHEMBL5271300)
Affinity DataEC50:  61nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  70nMAssay Description:Transactivation of mouse PPARdelta by cell-based luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  71nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  71nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50312471(2-(4-((4-(4-Morpholinophenyl)-5-(4-biphenyl)thiazo...)
Affinity DataEC50:  72nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  76nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  76nMMore data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM28661(2-{2-methyl-4-[({4-methyl-2-[4-(trifluoromethyl)ph...)
Affinity DataEC50:  77nMAssay Description:Agonist activity at mouse PPARdelta by FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50615965(CHEMBL5279568)
Affinity DataEC50:  79nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
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