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Compile Data Set for Download or QSAR

Found 2 hits of ec50 data for polymerid = 50006568   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Proteasome subunit beta type-7


(Homo sapiens)
BDBM50010992
PNG
(CHEMBL3259883)
Show SMILES CC(=O)Nc1cccc(c1)-c1nsc(=O)o1
Show InChI InChI=1S/C10H8N2O3S/c1-6(13)11-8-4-2-3-7(5-8)9-12-16-10(14)15-9/h2-5H,1H3,(H,11,13)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
AffyNet 
Article
n/an/an/an/a 4.20E+3n/an/an/an/a


TBA

Assay Description
Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...


Citation and Details
More data for this
Ligand-Target Pair
Proteasome subunit beta type-7


(Homo sapiens)
BDBM50010987
PNG
(CHEMBL3259880)
Show SMILES CC(=O)N[C@H](Cc1ccccc1)C(=O)Nc1ccc(cc1)-c1nsc(=O)o1
Show InChI InChI=1S/C19H17N3O4S/c1-12(23)20-16(11-13-5-3-2-4-6-13)17(24)21-15-9-7-14(8-10-15)18-22-27-19(25)26-18/h2-10,16H,11H2,1H3,(H,20,23)(H,21,24)/t16-/m1/s1
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
antibodypedia
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem

Similars

AffyNet 
Article
n/an/an/an/a 1.54E+4n/an/an/an/a


TBA

Assay Description
Inhibition of chymotrypsin-like activity of 26S proteasome in intact human Karpas 1106p cells assessed as substrate hydrolysis using Suc-LLVY-(D)-ami...


Citation and Details
More data for this
Ligand-Target Pair