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Compile Data Set for Download or QSAR

Found 23 hits of ec50 data for polymerid = 50006582,50006708,50006709,50006900,50006937,50006938,7093,7239   
Target
(Institution)
LigandTarget
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150818
PNG
(CHEMBL3774575)
Show SMILES CCCOc1cc(OCCCCN(C)C)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2ccc(OC)c(OC)c2)c1
PDB

KEGG

UniProtKB/SwissProt

GoogleScholar
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PC sid
PDB
UniChem

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PDB
Article
PubMed
n/an/an/an/a 50n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150820
PNG
(CHEMBL3774933)
Show SMILES CCCOc1cc(OCCCCN)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2ccc(OC)c(OC)c2)c1
PDB

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UniProtKB/SwissProt

GoogleScholar
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UniChem

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Article
PubMed
n/an/an/an/a 59n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150822
PNG
(CHEMBL3775348)
Show SMILES CCCOc1cc(OCCCCCN)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)cn2)c1
PDB

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UniProtKB/SwissProt

GoogleScholar
AffyNet 
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PC sid
UniChem

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Article
PubMed
n/an/an/an/a 110n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150821
PNG
(CHEMBL3775251)
Show SMILES CCCOc1cc(OCCCCN)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)cn2)c1
PDB

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UniProtKB/SwissProt

GoogleScholar
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UniChem

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Article
PubMed
n/an/an/an/a 120n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150819
PNG
(CHEMBL3774542)
Show SMILES CCCOc1cc(OCCCN)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2ccc(OC)c(OC)c2)c1
PDB

KEGG

UniProtKB/SwissProt

GoogleScholar
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PC sid
UniChem

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Article
PubMed
n/an/an/an/a 120n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150756
PNG
(CHEMBL3774766)
Show SMILES CCCOc1cc(OCCCCCCN)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2ccc(OC)c(OC)c2)c1
PDB

KEGG

UniProtKB/SwissProt

GoogleScholar
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CHEMBL
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Article
PubMed
n/an/an/an/a 170n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150758
PNG
(CHEMBL3775901)
Show SMILES CCCOc1cc(OCCCCCCN)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)cn2)c1
PDB

KEGG

UniProtKB/SwissProt

GoogleScholar
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CHEMBL
PC cid
PC sid
UniChem

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Article
PubMed
n/an/an/an/a 170n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150812
PNG
(CHEMBL3775853)
Show SMILES CCCOc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2ccc(OC)c(OC)c2)c1
PDB

KEGG

UniProtKB/SwissProt

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PDB
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Article
PubMed
n/an/an/an/a 830n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150811
PNG
(CHEMBL3775073)
Show SMILES CCCOc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)c(C)n2)c1
PDB

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PubMed
n/an/an/an/a 950n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150808
PNG
(CHEMBL3774507)
Show SMILES CC(C)COc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)c(C)n2)c1
PDB

KEGG

UniProtKB/SwissProt

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CHEMBL
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PDB
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PDB
Article
PubMed
n/an/an/an/a 1.30E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150757
PNG
(CHEMBL3774770)
Show SMILES CCCOc1cc(OCCCCCCO)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)cn2)c1
PDB

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UniProtKB/SwissProt

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CHEMBL
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Article
PubMed
n/an/an/an/a 1.80E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150761
PNG
(CHEMBL3775689)
Show SMILES Cn1cnc(c1)S(=O)(=O)Nc1cc2n(C)c(=O)n(C)c2cc1Oc1cccc(OCC2CCOC2)c1
PDB

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Article
PubMed
n/an/an/an/a 1.90E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150813
PNG
(CHEMBL3774653)
Show SMILES CCOc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)c(C)n2)c1
PDB

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PubMed
n/an/an/an/a 2.30E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150796
PNG
(CHEMBL3774529)
Show SMILES COCCCOc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)c(C)n2)c1
PDB

KEGG

UniProtKB/SwissProt

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Article
PubMed
n/an/an/an/a 2.70E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150803
PNG
(CHEMBL3774452)
Show SMILES CCCCOc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)c(C)n2)c1
PDB

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UniProtKB/SwissProt

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CHEMBL
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Article
PubMed
n/an/an/an/a 3.00E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150760
PNG
(CHEMBL3774883)
Show SMILES COc1ccc(cc1OC)S(=O)(=O)Nc1cc2n(C)c(=O)n(C)c2cc1Oc1cccc(OCCCCN(C)C)c1
PDB

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UniProtKB/SwissProt

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CHEMBL
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PubMed
n/an/an/an/a 3.20E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150815
PNG
(CHEMBL3775263)
Show SMILES COc1ccc(cc1OC)S(=O)(=O)Nc1cc2n(C)c(=O)n(C)c2cc1Oc1cccc(OCc2ccccc2)c1
PDB

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PubMed
n/an/an/an/a 3.90E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
3D
3D Structure (crystal)
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150814
PNG
(CHEMBL3775640)
Show SMILES Cc1nc(cn1C)S(=O)(=O)Nc1cc2n(C)c(=O)n(C)c2cc1Oc1cccc(OCc2ccccc2)c1
PDB

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PubMed
n/an/an/an/a 4.90E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150801
PNG
(CHEMBL3775132)
Show SMILES CC(C)COc1cccc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)C2CC2)c1
PDB

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PubMed
n/an/an/an/a 5.00E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150759
PNG
(CHEMBL3774638)
Show SMILES CCCOc1cc(OCCCCCCNC(=O)OC(C)(C)C)cc(Oc2cc3n(C)c(=O)n(C)c3cc2NS(=O)(=O)c2cn(C)cn2)c1
PDB

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UniProtKB/SwissProt

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CHEMBL
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PubMed
n/an/an/an/a 5.50E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150816
PNG
(CHEMBL3775286)
Show SMILES Cn1cnc(c1)S(=O)(=O)Nc1cc2n(C)c(=O)n(C)c2cc1Oc1cccc(OCc2ccccc2)c1
PDB

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UniProtKB/SwissProt

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PubMed
n/an/an/an/a 6.20E+3n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150817
PNG
(CHEMBL3774616)
Show SMILES Cn1cnc(c1)S(=O)(=O)Nc1cc2n(C)c(=O)n(C)c2cc1Oc1ccc(OCc2ccccc2)cc1
PDB

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UniProtKB/SwissProt

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UniChem

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PubMed
n/an/an/an/a>3.30E+4n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair
Transcription intermediary factor 1-alpha


(Homo sapiens)
BDBM50150800
PNG
(CHEMBL3775687)
Show SMILES CC(C)COc1cccc(Oc2ccc3n(C)c(=O)n(C)c3c2)c1
PDB

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UniProtKB/SwissProt

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CHEMBL
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PubMed
n/an/an/an/a>3.60E+4n/an/an/an/a



The University of Texas MD Anderson Cancer Center

Curated by ChEMBL


Assay Description
Inhibition of Flag-tagged TRIM24-PHD/bromodomain (unknown origin) expressed in human HeLa cells for 2 hrs by AlphaLisa assay


Citation and Details
More data for this
Ligand-Target Pair