Compile Data Set for Download or QSAR
maximum 50k data
Found 37 of ic50 data for polymerid = 50000579,50002909
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098915((R)-1-tert-Butyl-3-(4-methoxy-benzenesulfonyl)-6-o...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170292((S)-2-{4'-[(5-Methanesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  0.430nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170302((S)-2-{4'-[(5-Chloro-benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  0.600nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170287((S)-2-{4'-[(5-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  0.660nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170300((S)-3-Methyl-2-{4'-[(5-nitro-benzofuran-2-carbonyl...)
Affinity DataIC50:  0.700nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098924((R)-1-Cyclohexyl-3-(4-methoxy-benzenesulfonyl)-6-o...)
Affinity DataIC50:  0.75nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098913((R)-1,4-Bis-(4-methoxy-benzenesulfonyl)-[1,4]diaze...)
Affinity DataIC50:  0.840nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170294((S)-2-{4'-[(5-Acetylamino-benzofuran-2-carbonyl)-a...)
Affinity DataIC50:  0.980nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM28485((2S)-2-({4-[4-(1-benzofuran-2-amido)phenyl]benzene...)
Affinity DataIC50:  1.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170304((S)-2-{4'-[(5-Amino-benzofuran-2-carbonyl)-amino]-...)
Affinity DataIC50:  1.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098919((R)-1-Isopropyl-4-(4-methoxy-benzenesulfonyl)-7-ox...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098923((3R,9aS)-2-(4-Methoxy-benzenesulfonyl)-5-oxo-octah...)
Affinity DataIC50:  2nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098914((R)-5-Hydroxycarbamoyl-4-(4-methoxy-benzenesulfony...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170289((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  2.20nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170298((S)-2-{4'-[(4-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  2.30nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098920((R)-4-(4-Methoxy-benzenesulfonyl)-1-(1-methyl-1H-i...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170295((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098918((R)-1-Benzyl-3-(4-methoxy-benzenesulfonyl)-6-oxo-h...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098917((R)-1-Isopropyl-3-(4-methoxy-benzenesulfonyl)-6-ox...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170288((S)-2-{4'-[(5-Benzenesulfonylamino-benzofuran-2-ca...)
Affinity DataIC50:  3.40nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170296((S)-2-{4'-[(4-Benzyloxy-benzofuran-2-carbonyl)-ami...)
Affinity DataIC50:  3.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM8465((2R)-N-hydroxy-2-[(4-methoxybenzene)(pyridin-3-ylm...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM8465((2R)-N-hydroxy-2-[(4-methoxybenzene)(pyridin-3-ylm...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of rat matrix metalloprotease 13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170286((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170301((S)-2-{4'-[(Benzofuran-2-ylmethyl)-amino]-biphenyl...)
Affinity DataIC50:  4.90nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50291979(CHEMBL176602 | N-[[2-METHYL-4-HYDROXYCARBAMOYL]BUT...)
Affinity DataIC50:  7.40nMAssay Description:Inhibition of rat matrix metalloprotease 13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50098922((R)-3-(4-Methoxy-benzenesulfonyl)-1-methyl-6-oxo-h...)
Affinity DataIC50:  7.90nMAssay Description:Inhibition of Matrix metalloprotease-13More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170305((S)-2-{4'-[(Benzofuran-2-carbonyl)-amino]-biphenyl...)
Affinity DataIC50:  8.10nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170299((S)-3-Methyl-2-{4'-[([1,2,3]thiadiazole-4-carbonyl...)
Affinity DataIC50:  11nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170303((S)-2-[4'-(3-Methoxy-benzoylamino)-biphenyl-4-sulf...)
Affinity DataIC50:  14nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170293((S)-2-(4'-{[4-(1-Carboxy-ethoxy)-benzofuran-2-carb...)
Affinity DataIC50:  15nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170291((S)-2-{4'-[(7-Methoxy-benzofuran-2-carbonyl)-amino...)
Affinity DataIC50:  20nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170290(CHEMBL189955 | {4'-[(Benzofuran-2-carbonyl)-amino]...)
Affinity DataIC50:  22nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50170297((S)-2-{4'-[(1H-Indole-2-carbonyl)-amino]-biphenyl-...)
Affinity DataIC50:  35nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149234(Benzofuran-2-carboxylic acid (4-morpholin-4-yl-but...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Rattus norvegicus)
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194279(4-(2-(4-(4-(5-(2-methoxyethyl)-2,4,6-trioxo-hexahy...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of MMP13 in rat plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Bos taurus)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50149216(Benzofuran-2-carboxylic acid (2-{4-[benzyl-(2-hydr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory concentration against MMP-13 of bovine articular cartilage explantsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed