Compile Data Set for Download or QSAR
maximum 50k data
Found 40 of ic50 data for polymerid = 50001456
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063047(CHEMBL3398148)
Affinity DataIC50:  220nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063053(CHEMBL3398164)
Affinity DataIC50:  310nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50084637(2,2-Dimethyl-propionic acid 4-[2-(carboxymethyl-ca...)
Affinity DataIC50:  340nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063050(CHEMBL3398145)
Affinity DataIC50:  360nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063052(CHEMBL3398143)
Affinity DataIC50:  470nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101988(CHEMBL3398153)
Affinity DataIC50:  530nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataIC50:  530nMAssay Description:Inhibition of human PR3 using keto-D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM166437(US9073833, 5)
Affinity DataIC50:  610nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063054(CHEMBL3398165)
Affinity DataIC50:  610nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063051(CHEMBL3398144)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50384111(CHEMBL2029556)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101980(CHEMBL3398150)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50031630(CHEMBL3359765)
Affinity DataIC50:  1.91E+3nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063048(CHEMBL3398147)
Affinity DataIC50:  2.05E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101989(CHEMBL3398154)
Affinity DataIC50:  2.05E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063049(CHEMBL3398146)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM166438(US9073833, 6)
Affinity DataIC50:  2.37E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50063046(CHEMBL3398149)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101983(CHEMBL3398155)
Affinity DataIC50:  3.02E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101984(CHEMBL3398156)
Affinity DataIC50:  3.91E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101978(CHEMBL3398160)
Affinity DataIC50:  4.94E+3nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50384104(CHEMBL2029559)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50444297(CHEMBL3093815)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101977(CHEMBL3398159)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101985(CHEMBL3398157)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101981(CHEMBL3398161)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101982(CHEMBL3398162)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101987(CHEMBL3398163)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50101986(CHEMBL3398158)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Pr3 (unknown origin) using t-butyloxycarbonyl-Ala-Ala-Nva-thiobenzyl ester as substrate measured for 180 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50031631(CHEMBL3359767)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50384108(CHEMBL2029554)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50384112(CHEMBL2029557)
Affinity DataIC50:  1.45E+4nMAssay Description:Inhibition of proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate after 60 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50171289(Benzenemethanesulfonyl fluoride | CHEMBL190503 | P...)
Affinity DataIC50:  1.92E+4nMAssay Description:Inhibition of human PR3 using D-DY-FRET as substrate after 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50444296(CHEMBL3093814)
Affinity DataIC50:  4.75E+4nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50270029(2-Amino-N-[(S)-3-diazo-1-(4-iodo-benzyl)-2-oxo-pro...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of proteinase-3 in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50310690(CHEMBL1078411 | Cis-(S)-2-amino-N-((1R,2R)-1-cyano...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human Proteinase-3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50270040((S)-1-((1R,2R)-1-cyano-2-phenylcyclopropylamino)-1...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of proteinase-3 in human U937 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50260049(CHEMBL4104474)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of human neutrophil proteinase 3 using M4765 as substrate preincubated for 5 mins followed by substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50444295(CHEMBL3093806)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMyeloblastin(Homo sapiens (Human))
Chang Gung University

Curated by ChEMBL
LigandPNGBDBM50084637(2,2-Dimethyl-propionic acid 4-[2-(carboxymethyl-ca...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human proteinase 3 using N-MeOSuc-Ala-Ala-Pro-Val-p-nitroanilide as substrate measured for 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed