TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 3.60nMAssay Description:Displacement of [125I]eotaxin from BALB/c mouse CCR3 expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Antagonist activity at CCR3 assessed as eotaxin-induced chemotaxis in BALB/c mouse eosinophilsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of eotaxin-induced chemotaxis of mouse eosinophilsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of eotaxin-induced chemotaxis of mouse eosinophilsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Antagonist activity at CCR3 receptor in mouse eosinophil assessed as as inhibition of chemotaxisMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Inhibition of eotaxin-induced chemotaxis of mouse eosinophilsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 41nMAssay Description:Antagonist activity at CCR3 assessed as eotaxin-induced chemotaxis in BALB/c mouse eosinophilsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Displacement of [125I]eotaxin from BALB/c mouse CCR3 expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibition of mouse CCR3More data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 350nMAssay Description:Inhibitory activity against I-Eotaxin induced [Ca2+] response in mouse CCR3 receptorMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibitory activity against I-Eotaxin alpha binding to mouse CCR3 receptorsMore data for this Ligand-Target Pair
TargetProbable C-C chemokine receptor type 3(Mus musculus)
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Bristol-Myers Squibb Pharmaceutical Research Institute
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of mouse CCR3More data for this Ligand-Target Pair