Affinity DataIC50: 0.0670nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in absence of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0756nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in absence of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0763nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in presence of 100 uM of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0840nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in presence of 100 uM of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0929nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in absence of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0981nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in presence of 100 uM of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.520nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.620nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.860nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR assessed as GTP shiftMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Concentration required for 50% inhibition of [3H]-CHA binding on rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR assessed as GTP shiftMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR assessed as GTP shiftMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR assessed as GTP shiftMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity towards the adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Potency against rat brain A1 adenosine receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Evaluated for the binding affinity towards the Adenosine A1 receptor in cerebral cortices of Sprague-Dawley male rats using [3H]CHA as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes without NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Potency against rat brain adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membrane preparations using N6-[3H]-cyclohexyladenosine as a radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 3.10nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in presence of 100 uM of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.20nMAssay Description:Displacement of [3H]DPCPX from rat brain cortical membrane A1AR in absence of GTP by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Binding affinity to adenosine A1 receptor of rat brain membranes with 1 M NaCl by inhibition of [125-I]-labeled aminobenzyl adenosine bindingMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60nMAssay Description:Inhibitory activity against Adenosine A1 Receptor using [3H]-CHA in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Evaluated for binding affinity against Adenosine A1 receptorChecked by AuthorMore data for this Ligand-Target Pair