Affinity DataKd: 0.5nMAssay Description:Binding affinity to human CB1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.770nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 0.860nMAssay Description:Displacement of [3H]CP55940 from CB1 receptor in mouse brain at 100 nMMore data for this Ligand-Target Pair
Affinity DataKd: 0.860nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 1.20nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 1.25nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 1.25nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.40nMAssay Description:Displacement of [3H]CP55,940 from human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 1.66nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 1.80nMpH: 7.4Assay Description:Briefly, ~5μg of membranes were incubated at 30 °C for 60 min with [3H]CP55940 (147.9 Ci/mmol; PerkinElmer Life Sciences) or [3H]SR141716A (43 C...More data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Displacement of [3H]SR141716 from human CB1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 2.10nMpH: 7.4Assay Description:Briefly, ~5μg of membranes were incubated at 30 °C for 60 min with [3H]CP55940 (147.9 Ci/mmol; PerkinElmer Life Sciences) or [3H]SR141716A (43 C...More data for this Ligand-Target Pair
Affinity DataKd: 3.19nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 3.36nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 3.56nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 3.70nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 3.95nMAssay Description:Binding affinity to human CB1 receptor expressed in CHO cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 4.60nMAssay Description:Displacement of [3H]-SR-141716 from human CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 4.70nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1)More data for this Ligand-Target Pair
Affinity DataKd: 4.90nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1)More data for this Ligand-Target Pair
Affinity DataKd: 5.34nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 9nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 11nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 11.5nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 12.4nMAssay Description:Displacement of [3H]-SR-141716 from rat CB1 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 16.7nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 20.9nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 29.1nMAssay Description:Binding affinity to rat brain CB1 receptor after 90 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKd: 31nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 36nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 45nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 53.7nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 104nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 143nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 189nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 307nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 367nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 448nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 460nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 731nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Tested for binding affinity against Cannabinoid receptor 1 (CB1).More data for this Ligand-Target Pair
Affinity DataKd: 3.17E+3nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity against Cannabinoid receptor 1.More data for this Ligand-Target Pair