Affinity DataKd: 4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataIC50: 8nM Kd: 25nMAssay Description:Biochemical binding assays (DiscoveRx) and in vitro enzyme inhibition assays (LanthaScreen, Life Technologies) were conducted to determine the bindin...More data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 75nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 75nMAssay Description:Binding affinity to ACVR1More data for this Ligand-Target Pair
Affinity DataKd: 140nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 160nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 330nMAssay Description:Binding affinity to human ALK2 by KdELECT assayMore data for this Ligand-Target Pair
Affinity DataKd: 390nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 440nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 470nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 470nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 470nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 600nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 620nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 640nMAssay Description:Binding affinity to human ALK2 by KdELECT assayMore data for this Ligand-Target Pair
Affinity DataKd: 1.00E+3nMAssay Description:Binding affinity to human wild type partial length ACVR1 (C188 to C509 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.30E+3nMAssay Description:Binding affinity to human wild type partial length ACVR1 (C188 to C509 residues) expressed in bacterial expression system by Kinomescan methodMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.90E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Binding affinity to ACVR1More data for this Ligand-Target Pair
Affinity DataKd: 2.50E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 3.40E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 4.80E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 5.90E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 5.90E+3nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for ACVR1 kinase domainMore data for this Ligand-Target Pair