Affinity DataKd: 0.240nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
Affinity DataKd: 0.708nMAssay Description:Competitive antagonist activity at beta2-adrenoreceptor in guinea pig tracheal ring in the presence of N-(5-((1R)-2-(4-(4-(3,4-dimethoxyphenol)-1-oxo...More data for this Ligand-Target Pair
Affinity DataKd: 1.26nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 1.26nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 1.26nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 1.26nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 2.14nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 3.02nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
Affinity DataKd: 3.39nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 3.39nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 5.10nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring at basal tone assessed as bronchorelaxation activityMore data for this Ligand-Target Pair
Affinity DataKd: 6.31nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 7.94nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 8.91nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 8.91nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
Affinity DataKd: 9.55nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 12.6nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 15.8nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 16.6nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 18nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against histamine-induced co...More data for this Ligand-Target Pair
Affinity DataKd: 20.9nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 22.4nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 22.4nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 22.9nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring at basal tone assessed as bronchorelaxation activityMore data for this Ligand-Target Pair
Affinity DataKd: 28nMAssay Description:Agonist activity at adrenergic beta2 receptor in Hartley guinea pig tracheal ring assessed as bronchorelaxation activity against histamine-induced co...More data for this Ligand-Target Pair
Affinity DataKd: 30.2nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 32.4nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 32.4nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 33.1nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
Affinity DataKd: 39.8nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 39.8nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 39.8nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 39.8nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 43.6nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataKd: 47.9nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 50.1nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 57.5nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair
Affinity DataKd: 63.1nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 79.4nMAssay Description:Ability to block Beta-2 adrenergic receptor in guinea pig trachea preparationMore data for this Ligand-Target Pair
Affinity DataKd: 81.3nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 81.3nMAssay Description:The apparent pA2 value was measured for beta-2 adrenergic blocking activity on the trachea of guinea pigMore data for this Ligand-Target Pair
Affinity DataKd: 81.3nMAssay Description:Antagonist activity of compound against Beta-2 adrenergic receptor in isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataKd: 97.7nMAssay Description:Beta-2 adrenergic receptor blocking activity in trachea of guinea pig.More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:In vitro ability to block beta-2 adrenergic receptor in guinea pig trachea.More data for this Ligand-Target Pair
Affinity DataKd: 105nMAssay Description:In vitro beta-2 adrenergic receptor activity was determined by measuring inhibition of the isoproterenol induced relaxation in isolated guinea pig tr...More data for this Ligand-Target Pair