Compile Data Set for Download or QSAR
maximum 50k data
Found 29 of kd data for polymerid = 49000835,49000837
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500155(CHEMBL3747715)
Affinity DataKd:  0.0260nMAssay Description:Binding affinity to NPY1R in human SK-N-MC cells assessed as kinetically derived dissociation rate constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500155(CHEMBL3747715)
Affinity DataKd:  0.0400nMAssay Description:Binding affinity to NPY1R in human SK-N-MC cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500155(CHEMBL3747715)
Affinity DataKd:  0.0440nMAssay Description:Binding affinity to NPY1R in human SK-N-MC cells after 90 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500155(CHEMBL3747715)
Affinity DataKd:  0.0480nMAssay Description:Binding affinity to NPY1R in human SK-N-MC cells by Scatchard plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500155(CHEMBL3747715)
Affinity DataKd:  0.0740nMAssay Description:Binding affinity to NPY1R in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500155(CHEMBL3747715)
Affinity DataKd:  0.0830nMAssay Description:Binding affinity to NPY1R in human MCF7-Y1 cells by Scatchard plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500155(CHEMBL3747715)
Affinity DataKd:  0.140nMAssay Description:Binding affinity to NPY1R in human MCF7 cells after 90 mins by microbeta2 plate counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50246646((R)-Nalpha-(2,2-diphenylacetyl)-N-(4-hydroxybenzyl...)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to neuropeptide Y1 receptor in human SK-N-MC cells by kinetic experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50246646((R)-Nalpha-(2,2-diphenylacetyl)-N-(4-hydroxybenzyl...)
Affinity DataKd:  1.10nMAssay Description:Binding affinity to neuropeptide Y1 receptor in human MCF7 cells by kinetic experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50246646((R)-Nalpha-(2,2-diphenylacetyl)-N-(4-hydroxybenzyl...)
Affinity DataKd:  1.20nMAssay Description:Displacement of [3H]UR-MK114 from neuropeptide Y1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50246646((R)-Nalpha-(2,2-diphenylacetyl)-N-(4-hydroxybenzyl...)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to neuropeptide Y1 receptor in human SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50500164(CHEMBL3746028)
Affinity DataKd:  2nMAssay Description:Binding affinity to NPY1R in human SK-N-MC cells by liquid scintillation counting assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50060728((R)-2-(2,2-diphenylacetamido)-5-guanidino-N-(4-hyd...)
Affinity DataKd:  2.10nMAssay Description:Binding affinity to NPY1R in human SK-N-MC cells after 2 hrs by liquid scintillation counting assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50246646((R)-Nalpha-(2,2-diphenylacetyl)-N-(4-hydroxybenzyl...)
Affinity DataKd:  2.90nMAssay Description:Binding affinity to neuropeptide Y1 receptor in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50343728(3-((R)-9-Amino-4-(2,2-diphenylacetamido)-1-(4-hydr...)
Affinity DataKd:  5nMAssay Description:Binding affinity at Y1R in human MCF-7 cells by flowcytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003049(CHEMBL3559527 | Tyr-Pro-Ser-Lys-Pro-Ala-Asn-Pro-Gl...)
Affinity DataKd:  100nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003056(CHEMBL415353 | c(7,20)-Tyr-Pro-Ser-Lys-Pro-Asp-Glu...)
Affinity DataKd:  100nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50368404(CHEMBL409167)
Affinity DataKd:  780nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003045(CHEMBL425080 | c(30,34)-Ala-Arg-Tyr-Tyr-Ser-Ala-Le...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003054(CHEMBL406025 | c(30,34)-Ala-Arg-Tyr-Tyr-Ser-Ala-Le...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003043(CHEMBL437482 | c(2,30)Tyr-Glu-Ser-Lys-Pro-Ala-Leu-...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003055(CHEMBL414947 | Tyr-Pro-Ser-Lys-Pro-Ala-Leu-Arg-His...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003051(CHEMBL385339 | c(2,27)Tyr-Glu-Ser-Lys-Pro-Dpr-Leu-...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003052(CHEMBL413658 | c(33,36)-Ala-Arg-Tyr-Tyr-Ser-Ala-Le...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003048(CHEMBL265008 | Tyr-Pro-Ser-Lys-Pro-Lys-Leu-Arg-His...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003046(CHEMBL386202 | Tyr-Pro-Ala-His-Tyr-Ile-Asn-Leu-Ile...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003047(CHEMBL438211 | c(30,34)-Ala-Arg-Tyr-Tyr-Ser-Ala-Le...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003050(CHEMBL407742 | c(1,30)Glu-Pro-Ala-Tyr-Ile-Asn-Dpr-...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Cnrs/Ipbs (Institut De Pharmacologie Et Biologie Structurale)

Curated by ChEMBL
LigandPNGBDBM50003053(CHEMBL265637 | Tyr-Pro-Ser-Lys-Pro-Lys-Leu-Arg-His...)
Affinity DataKd: >1.00E+3nMAssay Description:Displacement of l25I-PYY from Neuropeptide Y receptor type 1 of human neuroblastoma SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed