TargetDual specificity mitogen-activated protein kinase kinase 4(Mus musculus)
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Affinity DataKd: 0.850nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Mus musculus)
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Affinity DataKd: 1.10nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.5nMAssay Description:Binding affinity to wild-type human partial length MKK4 (S84 to D399 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.70nMAssay Description:Binding affinity to wild-type human partial length MKK4 (S84 to D399 residues) expressed in mammalian expression system by Kinomescan methodMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Mus musculus)
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Affinity DataKd: 3.5nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 3.80nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 3.80nMAssay Description:Binding affinity to MEK4More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Mus musculus)
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Eberhard Karls Universit£T T£Bingen
Curated by ChEMBL
Affinity DataKd: 8.20nMAssay Description:Binding affinity to GST tagged mouse MKK4 expressed in Escherichia coli expression system measured by Kinomescan assayMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 70nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 70nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 70nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 150nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 250nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 330nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 390nMAssay Description:Binding affinity to MEK4 (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 590nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 590nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 590nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 630nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 630nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 700nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 810nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 910nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 930nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 930nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 930nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 1.80E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 2.30E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 3.40E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 3.70E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 4.00E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 4.80E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 4.80E+3nMAssay Description:Binding affinity to MEK4More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 4.80E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 4.80E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 5.50E+3nMAssay Description:Kd: For most assays, kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase an...More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: 9.90E+3nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MEK4More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MEK4More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MEK4More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MEK4More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to MEK4More data for this Ligand-Target Pair
TargetDual specificity mitogen-activated protein kinase kinase 4(Homo sapiens (Human))
Eberhard Karls Universit£T
Curated by ChEMBL
Eberhard Karls Universit£T
Curated by ChEMBL
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for MEK4 kinase domainMore data for this Ligand-Target Pair