Compile Data Set for Download or QSAR
maximum 50k data
Found 12 of ki data for polymerid = 1043,1044
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM10440((5S)-5-[(12-{[(5S)-2-oxo-1,2,5,6,7,8-hexahydroquin...)
Affinity DataKi:  19.6nM ΔG°:  -43.6kJ/mole IC50:  52nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM10440((5S)-5-[(12-{[(5S)-2-oxo-1,2,5,6,7,8-hexahydroquin...)
Affinity DataKi:  20nMAssay Description:Inhibition of rat AChEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50342601(CHEMBL1255901 | Huperzine A)
Affinity DataKi:  24nMAssay Description:Compound was tested for its ability to inhibit acetylcholinesterase (AChE) in rat brain; 0.024-0.040 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM10441((+)-Huperzine A | (+/-)Huperzine A | (-)-Huperzine...)
Affinity DataKi:  47.1nM ΔG°:  -41.4kJ/mole IC50:  114nMpH: 7.0 T: 2°CAssay Description:The cholinesterase assays were performed using colorimetric method reported by Ellman. Enzyme activity was determined by measuring the absorbance at ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50429847(CHEMBL2338670)
Affinity DataKi:  279nMAssay Description:Inhibition of AChE in rat cortex using acetylthiocholine iodide as substrate by double Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50104605(13-Eth-(E)-ylidene-11-methyl-6-aza-tricyclo[7.3.1....)
Affinity DataKi:  2.00E+3nMAssay Description:Compound was tested for its ability to inhibit acetylcholinesterase (AChE) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataKi:  2.75E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE by Michaelis-Menten equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50026058(CHEMBL3335259)
Affinity DataKi:  4.58E+3nMAssay Description:Inhibition of Sprague-Dawley rat brain AChE using acetylthiocholin iodide as substrate by Michaelis-Menten equationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50104603(13-Eth-(Z)-ylidene-11-methyl-6-aza-tricyclo[7.3.1....)
Affinity DataKi:  1.23E+4nMAssay Description:Compound was tested for its ability to inhibit acetylcholinesterase (AChE) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50028409(CHEMBL285508 | Trimethyl-[3-(2-oxo-2lambda*5*-[1,3...)
Affinity DataKi:  3.10E+4nMpH: 7.0Assay Description:Inhibitory constant of the compound against rat brain acetylcholinesterase at pH 7.0More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Weizmann Institute Of Science

LigandPNGBDBM50104604(11-Methyl-6-aza-tricyclo[7.3.1.0*2,7*]trideca-2(7)...)
Affinity DataKi: >5.00E+5nMAssay Description:Compound was tested for its ability to inhibit acetylcholinesterase (AChE) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed