Compile Data Set for Download or QSAR
maximum 50k data
Found 71 of ki data for polymerid = 50000596
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298756((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298754((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298760(CHEMBL574766 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  3.60nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298738(CHEMBL583783 | benzyl(2S,5S,8S,11S,14S)-8-(3-amino...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298761(CHEMBL574788 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298757((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298762(CHEMBL574924 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  6.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298739(CHEMBL583784 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  7.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298740(CHEMBL574324 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  8.80nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298714(CHEMBL574925 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  11.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298715(CHEMBL575847 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  12.8nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298716(CHEMBL574792 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  13.1nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298741(CHEMBL574931 | benzyl(2S,5S,8S,11S,14S)-7-cyclohex...)
Affinity DataKi:  13.1nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298717(CHEMBL574845 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  13.7nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298742(CHEMBL583785 | benzyl(2S,5S,8S,11S,14S)-8-(2-amino...)
Affinity DataKi:  18.2nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298718(CHEMBL574926 | benzyl(2S,5S,8S,11S,14S)-11-((1H-im...)
Affinity DataKi:  18.6nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298743(CHEMBL573527 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  19.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298755((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  19.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298719(CHEMBL574851 | benzyl(2S,5S,8S,11S,14S)-11-(3-amin...)
Affinity DataKi:  21.8nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434151(CHEMBL2381666)
Affinity DataKi:  22nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434153(CHEMBL2381668)
Affinity DataKi:  24nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298753((3S,6S,9S,12R)-9-(3-amino-3-oxopropyl)-3,6-bis(hyd...)
Affinity DataKi:  25.3nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298744(CHEMBL573414 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  25.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298752((5S,8S,11S,14R)-11-(3-amino-3-oxopropyl)-5,8-bis(h...)
Affinity DataKi:  27.5nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298720(CHEMBL574861 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  29.4nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298721(CHEMBL574927 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi:  37.4nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298722(CHEMBL574868 | benzyl(2S,5S,8S,11S,14S)-11-(2-amin...)
Affinity DataKi:  41.9nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434152(CHEMBL2381665)
Affinity DataKi:  43nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298745(CHEMBL583786 | benzyl(2S,5S,8S,11S,14S)-14-formyl-...)
Affinity DataKi:  43.8nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298751((5S,8S,11S,14R)-11-(4-aminobutyl)-5,8-bis(hydroxym...)
Affinity DataKi:  48.4nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298724(CHEMBL574885 | benzyl(2S,5S,8S,11R,14S)-8-(4-amino...)
Affinity DataKi: >50nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298728(CHEMBL583571 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi: >50nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298725(CHEMBL574928 | benzyl(2S,5S,8S,11S,14S)-8,11-bis(4...)
Affinity DataKi: >50nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298758((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi: >50nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298723(CHEMBL574878 | benzyl(2S,5S,8S,14S)-8-(4-aminobuty...)
Affinity DataKi: >50nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298727(CHEMBL573261 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi: >50nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298726(CHEMBL574895 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi: >50nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434148(CHEMBL2381663)
Affinity DataKi:  52nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434147(CHEMBL2381661)
Affinity DataKi:  61nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434145(CHEMBL2381660)
Affinity DataKi:  64nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298759((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  65nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298759((5S,8S,11S,14S,17R)-11-(4-aminobutyl)-5,8-bis(hydr...)
Affinity DataKi:  65nMAssay Description:Inhibition of human KLK3 using Mu-SRKSQQY-AMC as substrate by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  72nMpH: 7.8Assay Description:Inhibition of PSA (unknown origin) in 50 mM TRIS.HCL and 100 mM NaCl buffer at pH 7.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  72nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434146(CHEMBL2381670)
Affinity DataKi:  73nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  75nMAssay Description:Inhibition of PSA (unknown origin) in RPMIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298729(CHEMBL574929 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi: >100nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298730(CHEMBL574923 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi: >100nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50298731(CHEMBL583572 | benzyl(2S,5S,8S,11S,14S)-8-(4-amino...)
Affinity DataKi: >100nMAssay Description:Inhibition of prostate-specific antigen assessed as substrate hydrolysis by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50434143(CHEMBL2381658)
Affinity DataKi:  102nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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