Compile Data Set for Download or QSAR
maximum 50k data
Found 41 of ki data for polymerid = 50007805
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459745(CHEMBL4210431)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606137(CHEMBL5187921)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataKi:  56nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459744(CHEMBL4204744)
Affinity DataKi:  63nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459731(CHEMBL4216416)
Affinity DataKi:  90nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459737(CHEMBL4211204)
Affinity DataKi:  101nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606139(CHEMBL5198951)
Affinity DataKi:  109nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606141(CHEMBL5187149)
Affinity DataKi:  112nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459727(CHEMBL4206834)
Affinity DataKi:  119nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459738(CHEMBL4209820)
Affinity DataKi:  150nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606142(CHEMBL5197715)
Affinity DataKi:  157nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606146(CHEMBL5206253)
Affinity DataKi:  184nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606144(CHEMBL5199592)
Affinity DataKi:  204nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606140(CHEMBL5184570)
Affinity DataKi:  209nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606138(CHEMBL5207031)
Affinity DataKi:  231nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606147(CHEMBL5203898)
Affinity DataKi:  232nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataKi:  240nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606145(CHEMBL5190103)
Affinity DataKi:  245nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50606143(CHEMBL5208460)
Affinity DataKi:  254nMAssay Description:Binding affinity to MBP-tagged human recombinant ENL (489 to 559 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459735(CHEMBL4216170)
Affinity DataKi:  287nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459747(CHEMBL4216933)
Affinity DataKi:  369nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459726(CHEMBL4211962)
Affinity DataKi:  417nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459733(CHEMBL4209508)
Affinity DataKi:  510nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459745(CHEMBL4210431)
Affinity DataKi:  1.01E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459743(CHEMBL4209087)
Affinity DataKi:  1.24E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459748(CHEMBL4213382)
Affinity DataKi:  1.34E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459722(CHEMBL4204545)
Affinity DataKi:  1.43E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459742(CHEMBL4204647)
Affinity DataKi:  1.88E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459736(CHEMBL4216206)
Affinity DataKi:  2.15E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459729(CHEMBL4217882)
Affinity DataKi:  2.35E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459739(CHEMBL4204942)
Affinity DataKi:  3.37E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459732(CHEMBL4206070)
Affinity DataKi:  3.44E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459740(CHEMBL4214833)
Affinity DataKi:  4.89E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459724(CHEMBL4217790)
Affinity DataKi:  6.29E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459746(CHEMBL4212941)
Affinity DataKi:  7.73E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459741(CHEMBL4209918)
Affinity DataKi:  8.04E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459734(CHEMBL4208554)
Affinity DataKi:  1.46E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459728(CHEMBL4205558)
Affinity DataKi:  1.52E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459721(CHEMBL4213487)
Affinity DataKi:  2.01E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459725(CHEMBL4204221)
Affinity DataKi:  6.02E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein ENL(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459723(CHEMBL4218308)
Affinity DataKi:  6.20E+4nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged ENL (unknown origin) (489 to 559 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed