Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Antagonist activity at human recombinant 5HT3 receptor assessed as inhibition of RAMH-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 1.60nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Antagonist activity at rat recombinant 5HT3 receptor assessed as inhibition of RAMH-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 2.40nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 2.70nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 3nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 3.80nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 4.20nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 4.20nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 6.60nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 6.90nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracell...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 7.20nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 9.20nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracell...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 9.5nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 12.6nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 14nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 14.5nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Activity at SER3 receptor expressed in HEK293 cells assessed as increase in calcium by calcium imaging assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 32nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 54nMAssay Description:Effective concentration against 5-Hydroxytryptamine 3 receptor by measuring [14C]-guanidinium uptake on NG108-15 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 141nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as decrease in 10 uM 5-chloroindole-induced increase in intracell...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
European Research Centre For Drug Discovery And Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery And Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Agonist activity at 5HT3 receptor in voltage-stimulated guinea pig left atrium assessed as positive inotropic potencyMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Partial agonist activity at human 5HT3A receptor expressed in HEK293 cells assessed as effect on serotonin-induced responseMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbacholMore data for this Ligand-Target Pair
Affinity DataEC50: 240nMAssay Description:Binding affinity of the compound against human 5-hydroxytryptamine 3A receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 320nMAssay Description:Agonist activity at human wild type 5-HT3A receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(GUINEA PIG)
European Research Centre For Drug Discovery And Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery And Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Intrinsic activity at 5HT3 receptor in voltage-stimulated guinea pig left atrium assessed as positive inotropic potency relative to serotoninMore data for this Ligand-Target Pair
Affinity DataEC50: 457nMAssay Description:Antagonist activity at human 5HT3A receptor expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 500nMAssay Description:Agonist activity at human wild type 5-HT3A/5-HT3B receptor expressed in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 800nMAssay Description:Agonist activity at wild type mouse 5HT3A receptor expressed in Xenopus oocyte by two-electrode voltage patch clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: 2.10E+3nMAssay Description:Agonist activity at human 5HT3A receptor expressed in xenopus oocytes by electrophysiological methodMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:Antagonist activity at human recombinant 5-HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Homo sapiens (Human))
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Universita' Degli Studi Di Salerno
Curated by ChEMBL
Affinity DataEC50: 2.80E+3nMAssay Description:Agonist activity at human 5-HT43AB receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40E+3nMAssay Description:Agonist activity at wild type mouse 5HT3A receptor expressed in Xenopus oocyte by two-electrode voltage patch clamp methodMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80E+3nMAssay Description:Agonist activity at human 5-HT43A receptor expressed in Xenopus laevis oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity at human recombinant 5-HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair