Compile Data Set for Download or QSAR
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Found 921 Enz. Inhib. hit(s) with Target = 'Bombesin receptor subtype-3'
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127518(CHEMBL57104 | peptidomimetic)
Affinity DataEC50:  0.190nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533323(CHEMBL4435571)
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533327(CHEMBL4461212)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533327(CHEMBL4461212)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447496(CHEMBL3115400)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50381914(CHEMBL2023109 | MK-7725)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127544(CHEMBL56369 | peptidomimetic)
Affinity DataEC50:  1.40nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127520(CHEMBL57438 | peptidomimetic)
Affinity DataEC50:  1.5nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447479(CHEMBL3115386)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447479(CHEMBL3115386)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447477(CHEMBL3115388)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447477(CHEMBL3115388)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533320(CHEMBL4580739)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533331(CHEMBL4448589)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533331(CHEMBL4448589)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533320(CHEMBL4580739)
Affinity DataEC50:  2nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127539(3-(1H-Indol-3-yl)-N-phenethyl-2-(2-phenylacetylami...)
Affinity DataEC50:  2.10nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127527(CHEMBL294647 | peptidomimetic)
Affinity DataEC50:  2.20nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(RAT)
TBA

Curated by ChEMBL
LigandPNGBDBM50336889((2S)-1,1,1-trifluoro-2-[4-(1H-pyrazol-1-yl)phenyl]...)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at rat BRS-3 expressed in HEK293AEQ cells assessed as induction of intracellular calcium mobilization by aequorin bioluminescence as...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447477(CHEMBL3115388)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447497(CHEMBL3115399)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447477(CHEMBL3115388)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447497(CHEMBL3115399)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50314969(2-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447492(CHEMBL3115373)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447492(CHEMBL3115373)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50316914(5-((4'-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)...)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at mouse BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127529(2-[2-(4-Chloro-benzylamino)-acetylamino]-3-(1H-ind...)
Affinity DataEC50:  2.90nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533320(CHEMBL4580739)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533320(CHEMBL4580739)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533327(CHEMBL4461212)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50533327(CHEMBL4461212)
Affinity DataEC50:  3nMAssay Description:Agonist activity at mouse BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533326(CHEMBL4593256)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50533326(CHEMBL4593256)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human BRS3 expressed in CHOK1 cells measured after 1 hrs by IP-One HTRF assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50314977(5-(4-(2-(4-(2,2-dimethylbutyl)-1H-imidazol-2-yl)et...)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293 cells coexpressing AEQ over 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50127547(CHEMBL57559 | peptidomimetic)
Affinity DataEC50:  3.10nMAssay Description:Effective concentration required against human bombesin receptor 3 (BRS-3) in CHO cells by using FLIPR assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447479(CHEMBL3115386)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447479(CHEMBL3115386)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Technische UniversitäT MüNchen

Curated by ChEMBL
LigandPNGBDBM50041425(CHEMBL3356412)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at human BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447499(CHEMBL3115397)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at mouse BRS-3 expressed in CHOK1 cells after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50447475(CHEMBL3115390)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at mouse BRS3 expressed in CHO-K1 cells by IP-One HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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