Affinity DataEC50: 1.40E+4nMAssay Description:Inhibition of Apaf-1-caspase 9-cytochrome c-caspase 3 complex in human HEK293 cytosolic extract using afc-DEVD as substrate preincubated for 30 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.44E+4nMAssay Description:Inhibition of Apaf-1-caspase 9-cytochrome c-caspase 3 complex in human HEK293 cytosolic extract using afc-DEVD as substrate preincubated for 30 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.68E+4nMAssay Description:Inhibition of Apaf-1-caspase 9-cytochrome c-caspase 3 complex in human HEK293 cytosolic extract using afc-DEVD as substrate preincubated for 30 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.70E+4nMAssay Description:Inhibition of Apaf-1-caspase 9-cytochrome c-caspase 3 complex in human HEK293 cytosolic extract using afc-DEVD as substrate preincubated for 30 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.39E+4nMAssay Description:Inhibition of Apaf-1-caspase 9-cytochrome c-caspase 3 complex in human HEK293 cytosolic extract using afc-DEVD as substrate preincubated for 30 mins ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.99E+4nMAssay Description:Inhibition of Apaf-1-caspase 9-cytochrome c-caspase 3 complex in human HEK293 cytosolic extract using afc-DEVD as substrate preincubated for 30 mins ...More data for this Ligand-Target Pair
Affinity DataKi: 9.46E+4nMAssay Description:Binding affinity to human recombinant COX-2 assessed as inhibition constant preincubated for 5 mins followed by arachidonic acid addition measured ev...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human recombinant cyclooxygenase 2More data for this Ligand-Target Pair
Affinity DataIC50: 9.62E+4nMAssay Description:Inhibition of ovine cyclooxygenase 1More data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of human recombinant cyclooxygenase 2More data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+5nMAssay Description:Inhibition of ovine cyclooxygenase 1More data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+3nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 85nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.59E+4nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 69nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
Affinity DataIC50: 2.44E+4nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
Affinity DataIC50: 6.56E+4nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
Affinity DataIC50: 1.34E+4nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
Affinity DataIC50: 2.43E+4nMAssay Description:Inhibition of sheep COX1More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit 2(Ovis aries)
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Shahid Beheshti University Of Medical Sciences
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of sheep COX2More data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit NDUFA4(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory concentration against NADH ubiquinone oxidoreductaseMore data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit NDUFA4(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibitory concentration against NADH ubiquinone oxidoreductaseMore data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit NDUFA4(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibitory concentration against NADH-ubiquinone oxidoreductaseMore data for this Ligand-Target Pair
TargetCytochrome c oxidase subunit NDUFA4(Homo sapiens (Human))
The Scripps Research Institute
Curated by ChEMBL
The Scripps Research Institute
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibitory concentration against NADH-ubiquinone oxidoreductaseMore data for this Ligand-Target Pair
Affinity DataIC50: 540nMAssay Description:Thromboxane (TXA2) receptor antagonist activity using human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Thromboxane (TXA2) receptor antagonist activity using human plateletMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataIC50: 610nMAssay Description:Antagonistic activity against TP-receptor by inhibition of U 46619-induced contraction of isolated guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production by ELISAMore data for this Ligand-Target Pair
Affinity DataKd: 950nMAssay Description:Binding affinity to Cytochrome CMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to Cytochrome CMore data for this Ligand-Target Pair
Affinity DataKd: 1.70E+4nMAssay Description:Binding affinity to Cytochrome CMore data for this Ligand-Target Pair