Found 318 Enz. Inhib. hit(s) with Target = 'G protein-activated inward rectifier potassium channel 1' TargetG protein-activated inward rectifier potassium channel 1(Rattus norvegicus)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Affinity DataEC50: 0.0372nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Rattus norvegicus)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Affinity DataEC50: 0.0614nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Rattus norvegicus)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Affinity DataEC50: 0.280nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Rattus norvegicus)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Affinity DataEC50: 0.856nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Rattus norvegicus)
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Vanderbilt Screening Center For Gpcrs, Ion Channels And Transporters
Curated by PubChem BioAssay
Affinity DataEC50: 1.49nMAssay Description:Assay Provider: Colleen Niswender Assay Provider Affliation: Vanderbilt University Grant Title: Measurement of GPCR-mediated thallium flux through GI...More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 64nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 65nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 81nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 84nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 88nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 91nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 96nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 111nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 116nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 116nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 117nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 129nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 132nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 133nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 137nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 146nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Activation of GIRK1/2 (unknown origin) by cell-based thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 163nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 165nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 175nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 176nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 183nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 183nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 187nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 187nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 190nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 210nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: >221nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 239nMAssay Description:Activation of GIRK1/2 channel (unknown origin) expressed in HEK293 cells incubated for 6 mins by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 241nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 270nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 271nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Activation of human GIRK1/2 expressed in HEK293 cells co-expressing rat mGlu8 by thallium flux assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 310nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 310nMAssay Description:Activation of GIRK1/2 (unknown origin) by thallium-flux based assayMore data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
TargetG protein-activated inward rectifier potassium channel 1(Homo sapiens (Human))
University Of Nebraska
Curated by ChEMBL
University Of Nebraska
Curated by ChEMBL
Affinity DataEC50: 350nMAssay Description:Activation of GIRK1/2 (unknown origin)More data for this Ligand-Target Pair
