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Found 136 Enz. Inhib. hit(s) with Target = 'Lutropin-choriogonadotropic hormone receptor'
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335467(5-amino-N-tert-butyl-2-(methylthio)-4-(3-(2-oxo-2-...)
Affinity DataEC50:  1nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335473(5-amino-4-(3-(2-((1-(2-(2-(2-azidoethoxy)ethoxy)et...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335468((R)-4-(3-(2-((1-(2-(4-((4-(1-acetyl-6-biphenyl-4-y...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206401(CHEMBL246321 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335474((S)-4-(3-(2-((1-(2-(4-((4-(1-acetyl-6-biphenyl-4-y...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335469((R)-4-(3-(2-((1-(2-(2-(4-((4-(1-acetyl-6-biphenyl-...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335478((S)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335470((R)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335472((R)-4-(3-(2-((1-(14-(4-((4-(1-acetyl-6-biphenyl-4-...)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335477((S)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...)
Affinity DataEC50:  57nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335471((R)-4-(3-(2-((1-(2-(2-(2-(2-(4-((4-(1-acetyl-6-bip...)
Affinity DataEC50:  61nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335476((S)-4-(3-(2-((1-(2-(2-(2-(4-((4-(1-acetyl-6-biphen...)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50335475((S)-4-(3-(2-((1-(2-(2-(4-((4-(1-acetyl-6-biphenyl-...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206398(CHEMBL429108 | N-(4-hydroxyphenethyl)-5-(1-(4-tert...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206402(CHEMBL439392 | N-((S)-1-amino-3-(3-hydroxyphenyl)-...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206399(CHEMBL247700 | N-((S)-2-amino-1-(4-hydroxyphenyl)-...)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206397((S)-N-(4-amino-4-oxo-1-phenylbutan-2-yl)-5-(1-(4-t...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189778(CHEMBL211405 | N-tert-butyl-5-amino-4-(3-methoxyph...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at LHCGR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206395((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189778(CHEMBL211405 | N-tert-butyl-5-amino-4-(3-methoxyph...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206400(CHEMBL247945 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189779(CHEMBL377399 | N-tert-butyl-5-amino-4-(3-methoxyph...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189775(CHEMBL377769 | N-tert-butyl-5-amino-4-(2,3-dimetho...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189776(CHEMBL211871 | tert-butyl 5-amino-4-(3-methoxyphen...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189777(CHEMBL212815 | N-tert-butyl-5-amino-4-(3-fluorophe...)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189773(CHEMBL211129 | N-tert-butyl-5-amino-4-(2-fluoro-3-...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50256858(CHEMBL474041 | Cyclopentyl-carbamic acid [1,1',3',...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human luteinizing hormone receptor expressed in CHOK1 cells assessed as c-AMP-mediated luciferase productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50189774(CHEMBL378091 | N-tert-butyl-5-amino-4-(3-hydroxyph...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at LHCGR expressed in HEK293 EM cells measured by intracellular cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206405((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206403(CHEMBL269261 | N-((S)-1-amino-3-(4-tert-butoxyphen...)
Affinity DataEC50:  1.21E+4nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50505787(CHEMBL4537998)
Affinity DataEC50: >1.60E+4nMAssay Description:Agonist activity at human luteinizing hormone receptor incubated for 60 mins by cell based TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206404((S)-N-(1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-y...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206396((S)-2-{3-[2-(4-tert-butyl-phenyl)-5-pyridin-3-yl-2...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50405789(CHEMBL412984)
Affinity DataKi:  0.0182nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230127(CHEMBL407606)
Affinity DataKi:  0.0245nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230129(CHEMBL407123)
Affinity DataKi:  0.0427nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230120(CHEMBL405737)
Affinity DataKi:  0.0776nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230123(CHEMBL385042)
Affinity DataKi:  0.0933nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230122(CHEMBL415571)
Affinity DataKi:  0.155nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230126(CHEMBL385468)
Affinity DataKi:  0.186nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230124(CHEMBL429240)
Affinity DataKi:  0.209nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50405770(CHEMBL216617)
Affinity DataKi:  0.282nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50206401(CHEMBL246321 | N-((S)-1-amino-3-(4-hydroxyphenyl)-...)
Affinity DataKi:  0.311nMAssay Description:Displacement of [125I]-hCG from LH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230128(CHEMBL437798)
Affinity DataKi:  0.380nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50405767(CHEMBL265413)
Affinity DataKi:  0.457nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50405769(CHEMBL275694)
Affinity DataKi:  0.525nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50405764(CHEMBL264298)
Affinity DataKi:  1.20nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50422274(GONADORELIN | Human gonadoliberin-i)
Affinity DataKi:  1.30nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50405782(CHEMBL413887)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLutropin-choriogonadotropic hormone receptor(Rattus norvegicus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50230130(CHEMBL266205)
Affinity DataKi:  1.40nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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