TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 34nMAssay Description:Inhibition of CBR1 (unknown origin)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 75nMAssay Description:Inhibition of CBR1 (unknown origin)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of CBR1 (unknown origin)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of CBR1 (unknown origin)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 270nMAssay Description:Inhibition of CBR1 (unknown origin)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of CBR1 (unknown origin)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of CBR1 (unknown origin)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 670nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 759nMAssay Description:Inhibition of CBR-mediated NADPH-dependent reduction of menadione to menadiolMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 788nMAssay Description:Inhibition of CBR-mediated NADPH-dependent reduction of menadione to menadiolMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity against high affinity component of Adenosine A1 receptor from rat brain membranes using [3H]-DPCPXMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3.27E+3nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 3.78E+3nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of recombinant human CBR1 using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of menadione from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.10E+4nMAssay Description:Displacement of daunorubicin from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.27E+4nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Displacement of daunorubicin from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Displacement of daunorubicin from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.15E+4nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 2.50E+4nMAssay Description:Displacement of daunorubicin from human recombinant CBR expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 40nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 520nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 600nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 2.03E+3nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair
TargetCarbonyl reductase [NADPH] 1(Homo sapiens (Human))
Gifu Pharmaceutical University
Curated by ChEMBL
Gifu Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 3.43E+3nMAssay Description:Binding affinity to human recombinant carbonyl reductase 1 expressed in Escherichia coli assessed as NADPH oxidation using isatin as substrateMore data for this Ligand-Target Pair