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Found 31 Enz. Inhib. hit(s) with Target = 'PBP2'
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50217404(CHEMBL348278)
Affinity DataIC50:  1.40nMAssay Description:Compound was tested for its binding affinity towards Penicillin-binding protein 2a (PBP2a) using [13H]-benzylpenicillinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50217406(CHEMBL351921)
Affinity DataIC50:  1.60nMAssay Description:Compound was tested for its binding affinity towards Penicillin-binding protein 2a (PBP2a) using [13H]-benzylpenicillinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50217407(CHEMBL161482)
Affinity DataIC50:  2.40nMAssay Description:Compound was tested for its binding affinity towards Penicillin-binding protein 2a (PBP2a) using [13H]-benzylpenicillinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50217403(CHEMBL161759)
Affinity DataIC50:  7.10nMAssay Description:Compound was tested for its binding affinity towards Penicillin-binding protein 2a (PBP2a) using [13H]-benzylpenicillinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50217402(CHEMBL157932)
Affinity DataIC50:  18nMAssay Description:Compound was tested for its binding affinity towards Penicillin-binding protein 2a (PBP2a) using [13H]-benzylpenicillinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50217405(CHEMBL159153)
Affinity DataIC50:  22nMAssay Description:Compound was tested for its binding affinity towards Penicillin-binding protein 2a (PBP2a) using [13H]-benzylpenicillinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213266(CHEBI:471744 | Imipenem | MK-0787)
Affinity DataIC50:  188nMAssay Description:Compound was tested for its binding affinity towards Penicillin-binding protein 2a (PBP2a) using [13H]-benzylpenicillinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213270(CHEMBL33235)
Affinity DataIC50:  649nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213260(CHEMBL34381)
Affinity DataIC50:  876nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213261(CHEMBL430547)
Affinity DataIC50:  1.35E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213265(CHEMBL287296)
Affinity DataIC50:  1.93E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213222(CHEMBL33794)
Affinity DataIC50:  2.08E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213262(CHEMBL286644)
Affinity DataIC50:  2.59E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213269(CHEMBL430721)
Affinity DataIC50:  2.76E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213220(CHEMBL30322)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213259(CHEMBL30991)
Affinity DataIC50:  3.36E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213268(CHEMBL410910)
Affinity DataIC50:  3.78E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213264(CHEMBL287558)
Affinity DataIC50:  3.82E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213254(CHEMBL287661)
Affinity DataIC50:  5.02E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213267(CHEMBL282600)
Affinity DataIC50:  6.24E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213219(CHEMBL33583)
Affinity DataIC50:  8.06E+3nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213263(CHEMBL284058)
Affinity DataIC50:  1.06E+4nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213218(CHEMBL283624)
Affinity DataIC50:  2.36E+4nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213221(CHEMBL282641)
Affinity DataIC50:  3.05E+4nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213253(CHEMBL285914)
Affinity DataIC50:  3.44E+4nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213255(CHEMBL33323)
Affinity DataIC50:  4.11E+4nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213256(CHEMBL284293)
Affinity DataIC50:  4.28E+4nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213271(CHEMBL33672)
Affinity DataIC50:  7.14E+4nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213257(CHEMBL34220)
Affinity DataIC50:  1.12E+5nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213258(CHEMBL30267)
Affinity DataIC50:  2.36E+5nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails
TargetPBP2A(Staphylococcus aureus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50213266(CHEBI:471744 | Imipenem | MK-0787)
Affinity DataIC50:  4.28E+5nMAssay Description:Binding affinity towards Penicillin-binding protein 2a from homogeneous MRSA COL strain using [3H]-radioligandMore data for this Ligand-Target Pair
In DepthDetails