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Found 40 Enz. Inhib. hit(s) with Target = 'Breast cancer type 1 susceptibility protein'
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345640((S)-2-((2S,3R)-2-((S)-1-((S)-2-acetamido-3-(phosph...)
Affinity DataKd:  190nMAssay Description:Binding affinity to BRCA1 by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345643(CHEMBL1784787)
Affinity DataKd:  410nMAssay Description:Binding affinity to BRCA1 by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345642((2S,5S,8S,11S,14S)-2-((S)-2-((2S,3R)-1-((S)-1-((S)...)
Affinity DataKd:  440nMAssay Description:Binding affinity to BRCA1 by isothermal titration calorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380359(CHEMBL2017822)
Affinity DataKi:  40nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380358(CHEMBL2017821)
Affinity DataKi:  80nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380353(CHEMBL2017816)
Affinity DataKi:  100nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380352(CHEMBL2017815)
Affinity DataKi:  130nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345641((S)-2-((S)-2-((S)-1-((S)-2-acetamido-3-(phosphonoo...)
Affinity DataKi:  200nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345640((S)-2-((2S,3R)-2-((S)-1-((S)-2-acetamido-3-(phosph...)
Affinity DataKi:  270nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380354(CHEMBL2017817)
Affinity DataKi:  500nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380351(CHEMBL2017814)
Affinity DataKi:  540nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380349(CHEMBL2017812)
Affinity DataKi:  1.24E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345623((S)-2-acetamido-3-((S)-2-((2S,3R)-1-((S)-1-amino-1...)
Affinity DataKi:  1.85E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345629((S)-2-acetamido-3-((S)-2-((S)-1-((S)-1-amino-1-oxo...)
Affinity DataKi:  1.96E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380357(CHEMBL2017820)
Affinity DataKi:  4.04E+3nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380355(CHEMBL2017818)
Affinity DataKi:  1.21E+4nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380356(CHEMBL2017819)
Affinity DataKi:  1.57E+4nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50380350(CHEMBL2017813)
Affinity DataKi:  1.94E+4nMAssay Description:Inhibition of BRCT domain of His-tagged BRCA1 after 1 min by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50221433(1-(9,10,10-trioxo-9,10-dihydro-10lambda*6*-thioxan...)
Affinity DataKi:  3.00E+4nMAssay Description:Inhibition of BRCA1 assessed as BRCT-BACH1 interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50221434(3-(4-benzyl-piperidin-1-yl)-10,10-dioxo-10H-10lamb...)
Affinity DataKi:  3.80E+4nMAssay Description:Inhibition of BRCA1 assessed as BRCT-BACH1 interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50221432(3-(4-methyl-piperidin-1-yl)-10,10-dioxo-10H-10lamb...)
Affinity DataKi:  3.90E+4nMAssay Description:Inhibition of BRCA1 assessed as BRCT-BACH1 interactionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345641((S)-2-((S)-2-((S)-1-((S)-2-acetamido-3-(phosphonoo...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345637((S)-2-acetamido-3-((S)-2-((S)-2-((S)-1-amino-1-oxo...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345636((S)-2-acetamido-3-((S)-1-((S)-1-((S)-1-amino-1-oxo...)
Affinity DataIC50:  9.84E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345635((S)-2-acetamido-3-((S)-2-((2S,3R)-1-((S)-1-amino-3...)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345634((2S)-2-acetamido-3-((2S)-2-((2S,3R)-1-(1-amino-3-(...)
Affinity DataIC50:  1.72E+5nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345633((2S)-2-acetamido-3-((2S)-2-((2S,3R)-1-(1-amino-3-(...)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345632((S)-2-acetamido-3-((S)-2-((S)-1-((S)-1-amino-1-oxo...)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345631((S)-2-acetamido-3-((S)-2-((2S,3S)-1-((S)-1-amino-1...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345630((S)-2-acetamido-3-((S)-2-((S)-1-((S)-1-amino-1-oxo...)
Affinity DataIC50:  3.01E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345629((S)-2-acetamido-3-((S)-2-((S)-1-((S)-1-amino-1-oxo...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345628((S)-2-acetamido-3-((S)-2-((S)-1-((S)-1-amino-1-oxo...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345627((S)-2-acetamido-3-((S)-1-((2S,3R)-1-((S)-1-amino-1...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345626((2R,3S)-3-acetamido-4-((S)-2-((2S,3R)-1-((S)-1-ami...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345625(2-((S)-2-acetamido-3-((S)-2-((2S,3R)-1-((S)-1-amin...)
Affinity DataIC50:  5.28E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345624((S)-4-acetamido-5-((S)-2-((2S,3R)-1-((S)-1-amino-1...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345623((S)-2-acetamido-3-((S)-2-((2S,3R)-1-((S)-1-amino-1...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345638((2R,5R,8R,11R)-11-benzyl-2-carbamoyl-8-((S)-1-hydr...)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345639((S)-2-amino-3-((S)-2-((2S,3R)-1-((S)-1-amino-1-oxo...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreast cancer type 1 susceptibility protein(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50345640((S)-2-((2S,3R)-2-((S)-1-((S)-2-acetamido-3-(phosph...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of BRCA1 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed