Affinity DataKd: 1.60E+3nMAssay Description:Dissociation constant of the copound at P2X purinoceptor 1 (P2X1) from rat vas deferens was reportedMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataKi: 49nMAssay Description:Competitive antagonist activity at human P2X4 receptor expressed in 1321N1 cell membrane assessed as inhibition of [35S]ATPgammaS binding by scintill...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of inward ion current elicited by ATP at rat P2X4 receptor (wild type)More data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of inward ion current elicited by ATP at rat P2X4 receptor (mutant type)More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: 2.75E+4nMAssay Description:Inhibition of inward ion current elicited by ATP at human P2X4 receptor (mutant type)More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at P2X4 receptor up to 10 uMMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of P2X4 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.19E+5nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 10 uMMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 500nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 1.50E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+5nMAssay Description:The compound was evaluated for antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
Affinity DataIC50: 9.60E+3nMAssay Description:The compound was evaluated for antagonist activity against P2X purinoceptor 1 (P2X1) receptor from rat vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.30E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+5nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 2.50E+4nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 7.40E+3nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) at 3 uM,expressed in Xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80E+4nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+4nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 1.00E+3nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 1.28E+5nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
Affinity DataEC50: 3.30E+4nMAssay Description:The compound was evaluated for antagonist activity against recombinant rat P2X purinoceptor 4 (P2X4) 3 uMMore data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataEC50: 490nMAssay Description:Antagonist activity against recombinant human P2X purinoceptor 4 (P2X4)More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: 1.46E+5nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: 7.28E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: 1.53E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: 5.14E+4nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair
TargetP2X purinoceptor 4(Homo sapiens (Human))
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Max-Planck Institute For Experimental Medicine
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human P2X4 receptor expressed in human 1321N1 cells assessed as inhibition of ATP-induced cytosolic calcium influx preincubate...More data for this Ligand-Target Pair