Compile Data Set for Download or QSAR
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Found 1643 Enz. Inhib. hit(s) with Target = 'Phospholipase A2'
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153280(1-Benzofuran-2-yl-3-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  4.52E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23759(3-{4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153282(1-Benzofuran-2-yl-3-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.27E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153283(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4-dimethy...)
Affinity DataIC50:  3.22E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153284(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(2,3-dimet...)
Affinity DataIC50:  2.28E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153285(1-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-3-(4,7-dimet...)
Affinity DataIC50:  1.91E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153286(3-Benzofuran-2-yl-5-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  3.54E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153287(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  2.11E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153288(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  9.17E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153289(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  2.22E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153290(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  1.92E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153291(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  7.12E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153292(3-Benzofuran-2-yl-5-(4-dimethylamino-naphthalen-1-...)
Affinity DataIC50:  2.22E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153293(3-Benzofuran-2-yl-5-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  1.46E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153294(3-Benzofuran-2-yl-5-(2,3-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  8.46E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153295(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4-dimethy...)
Affinity DataIC50:  1.72E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153296(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(2,3-dimet...)
Affinity DataIC50:  1.73E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153297(3-(2,3-Dihydro-benzo[1,4]dioxin-6-yl)-5-(4,7- dime...)
Affinity DataIC50:  5.12E+3nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  620nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23750(3-{4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}-4...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23752(3-{4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23753(3-{4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50:  5.08E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23754(3-({4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}m...)
Affinity DataIC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23755(3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50:  1.00E+4nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23756(3-({4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50:  2.20E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23757(3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23758(3-{4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23759(3-{4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50:  1.10E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23760(3-({4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl...)
Affinity DataIC50:  9.00E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23761(3-({4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50:  4.00E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23762(3-({4-[(4-octadecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50:  800nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23763(3-({4-[(4-icosylpiperazin-1-yl)carbonyl]phenyl}met...)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23764(3-({4-[(4-docosylpiperazin-1-yl)carbonyl]phenyl}me...)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23765(3-{[4-(4-tetradecylpiperazin-1-yl)phenyl]methyl}-4...)
Affinity DataIC50:  4.50E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23766(3-{[4-(4-hexadecylpiperazin-1-yl)phenyl]methyl}-4,...)
Affinity DataIC50:  3.50E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23767(3-{[4-(4-octadecylpiperazin-1-yl)phenyl]methyl}-4,...)
Affinity DataIC50:  2.71E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23768(3-(2-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phen...)
Affinity DataIC50:  1.87E+4nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23769(3-(3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phen...)
Affinity DataIC50:  5.30E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23770(3-{[4-(tetradecyloxy)phenyl]methyl}-4,5-dihydro-1,...)
Affinity DataIC50:  4.00E+3nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23771((3-{[1-benzyl-3-(carbamoylmethyl)-2-ethyl-1H-indol...)
Affinity DataIC50:  470nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23750(3-{4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}-4...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23752(3-{4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23753(3-{4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}-4,...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23754(3-({4-[(4-tetradecylpiperazin-1-yl)methyl]phenyl}m...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23755(3-({4-[(4-hexadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23756(3-({4-[(4-octadecylpiperazin-1-yl)methyl]phenyl}me...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23757(3-{4-[(4-tetradecylpiperazin-1-yl)carbonyl]phenyl}...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, major isoenzyme(Sus scrofa (pig))
Universite Paris 7-Denis Diderot

LigandPNGBDBM23758(3-{4-[(4-hexadecylpiperazin-1-yl)carbonyl]phenyl}-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:PLA2 activity is by using the fluorescent phospholipid analogue, beta-pyC-10-PG as the substrate. The increase in fluorescence (ex @342 nm and em@388...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2 group V(Homo sapiens (Human))
Universiti Kebangsaan Malaysia, Jalan Raja Muda Abdul Aziz

LigandPNGBDBM153281(1-Benzofuran-2-yl-3-(4,7-dimethoxy-naphthalen-1-yl...)
Affinity DataIC50:  2.78E+4nMpH: 7.5 T: 2°CAssay Description:Briefly, sn-2ester bond of the substrate 1,2-bis(heptanoylthio)-glycerophosphocholine was hydrolyzed by PLA2-V followed by the exposure of free thiol...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPhospholipase A2, membrane associated(Homo sapiens (Human))
Universite Paris 7-Denis Diderot

LigandPNGBDBM123738(DCSD 002847 (2))
Affinity DataIC50:  8.60E+3nMpH: 8.0Assay Description:The reaction mixture contained 160 uL of reaction buffer [50 mM Tris-HCl (pH 8.0), 100 mM NaCl, 5 ug/mL bovine serum albumin (BSA), 5 uM CaCl2, and 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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