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Found 67 Enz. Inhib. hit(s) with Target = 'Xaa-Pro dipeptidase'
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366413(PHOSPHOENOLPYRUVATE)
Affinity DataKi:  8.5nMpH: 6.0Assay Description:Inhibition of prolidase from swine kidney at a pH 6More data for this Ligand-Target Pair
In DepthDetails Article
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285931(2-((1R,2R)-2-Carboxy-cyclopentyl)-2-oxo-ethyl-ammo...)
Affinity DataKi:  270nMAssay Description:Inhibitory activity against porcine kidney prolidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50366413(PHOSPHOENOLPYRUVATE)
Affinity DataKi:  300nMAssay Description:Inhibitory constant for inhibition of prolidase in the first phase of biphasic inhibitionMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50240386(5-amino-4-oxopentanoic acid | 5-aminolevulinic aci...)
Affinity DataKi:  9.60E+5nMAssay Description:Inhibitory activity against porcine kidney prolidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285933(2-((1R,2R)-2-Carboxy-cyclohexyl)-2-oxo-ethyl-ammon...)
Affinity DataKi:  1.10E+6nMAssay Description:Inhibitory activity against porcine kidney prolidaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078391((S)-1-[(R)-3-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078397(1-(3-Amino-2-hydroxy-5-methyl-hexanoyl)-pyrrolidin...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50:  1.70E+6nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078401((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078400(1-[1-(3-Amino-2-hydroxy-4-phenyl-butyryl)-4-hydrox...)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+7nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078394((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078393((S)-1-[(S)-1-((2S,3R)-3-Amino-2-hydroxy-4-phenyl-b...)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078402((S)-1-((R)-3-Amino-2-hydroxy-5-methyl-hexanoyl)-py...)
Affinity DataIC50:  660nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078392((S)-1-((2R,3R)-3-Amino-2-hydroxy-5-methyl-hexanoyl...)
Affinity DataIC50:  4.10E+5nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078399((S)-1-((3R,4S)-4-Amino-3-hydroxy-6-methyl-heptanoy...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078398(2-[(S)-2-((S)-1-Carbamoyl-ethylcarbamoyl)-pyrrolid...)
Affinity DataIC50: >2.00E+6nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50078395((S)-1-(2-Hydroxycarbamoyl-cyclohexanecarbonyl)-pyr...)
Affinity DataIC50: >5.00E+7nMAssay Description:Inhibition against Prolidase from pig kidney.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50153382(CHEMBL183289 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50153386(CHEMBL435882 | Trifluoro-acetate1-(2-fluoro-benzyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50153384(CHEMBL364102 | Trifluoro-acetate3-{(S)-2-[4-((R)-1...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50153381(CHEMBL186482 | Trifluoro-acetate1-(2-fluoro-benzyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50153401(CHEMBL184346 | Trifluoro-acetate1-(2-fluoro-benzyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232507(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232512((2R)-4-[(8S)-8-(4-fluorobenzyl)-3-(trifluoromethyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232511((2R)-4-[8-ethyl-3-(trifluoromethyl)-5,6-dihydro[1,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232510((2R)-4-[8-benzyl-3-(trifluoromethyl)-5,6-dihydro[1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232505((2R)-4-[5,5-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM11162((1R)-3-oxo-3-[3-(trifluoroethyl)-5,6-dihydro[1,2,4...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232501((2R)-4-[8-(2-fluorobenzyl)-3-(trifluoromethyl)-5,6...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232524((2R)-4-[8,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232520((2R)-4-oxo-4-[3-(trifluoromethyl)-8-[2-(trifluorom...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232521((2R)-4-[(6R)-6-methyl-3-(trifluoromethyl)-5,6-dihy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232500(((2R)-4-[(6S)-6-methyl-3-(trifluoromethyl)-5,6-dih...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232508((2R)-4-[8-(2,2,2-trifluoroethyl)-3-(trifluoromethy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50371255(CHEMBL1203953)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232503((2R)-4-[8-(4-methoxybenzyl)-3-(trifluoromethyl)-5,...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232518((2R)-4-oxo-4-[8-(pyridin-2-ylmethyl)-3-(trifluorom...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232514((2R)-4-[8-allyl-3-(trifluoromethyl)-5,6-dihydro[[1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232520((2R)-4-oxo-4-[3-(trifluoromethyl)-8-[2-(trifluorom...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151819((R)-3-Amino-4-(2-fluoro-phenyl)-1-piperazin-1-yl-b...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232502((2R)-4-[(8S)-8-methyl-3-(trifluoromethyl)-5,6-dihy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232502((2R)-4-[(8S)-8-methyl-3-(trifluoromethyl)-5,6-dihy...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232510((2R)-4-[8-benzyl-3-(trifluoromethyl)-5,6-dihydro[1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232518((2R)-4-oxo-4-[8-(pyridin-2-ylmethyl)-3-(trifluorom...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232504((2R)-4-[5,8-dimethyl-3-(trifluoromethyl)-5,6-dihyd...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetXaa-Pro dipeptidase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50232506(2-[7-[(3R)-3-amino-4-(2,4,5-trifluorophenyl)butano...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of prolidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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