Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 9413
TargetProstacyclin receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464509(2-(((1s,4s)-4-((6-(4- methoxyphenyl)-3-oxo-5- phen...)
Affinity DataEC50:  8nMAssay Description:The HTRF® assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volum...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstacyclin receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464512(2-(((1s,4s)-4-((5-(3- chlorophenyl)-3-oxo-6- pheny...)
Affinity DataEC50:  73nMAssay Description:The HTRF® assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volum...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstacyclin receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464511(2-(((1s,4s)-4-((3-oxo-5,6-di- p-tolyl-1,2,4-triazi...)
Affinity DataEC50:  36nMAssay Description:The HTRF® assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volum...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstacyclin receptor(Homo sapiens (Human))
Arena Pharmaceuticals

US Patent
LigandPNGBDBM464510(2-(((1s,4s,)-4-((4-(3-chloro- 2-fluorophenyl)-6-ox...)
Affinity DataEC50:  31nMAssay Description:The HTRF® assay was carried out using a two-step protocol essentially according to the kit manufacturer's instructions, in 20 μL total volum...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent