Compile Data Set for Download or QSAR
maximum 50k data
Found 141 Enz. Inhib. hit(s) with all data for entry = 10308
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526635(1-acryloyl-N-(3-(((8-isopropyl-2-((1-methylpiperid...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526635(1-acryloyl-N-(3-(((8-isopropyl-2-((1-methylpiperid...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526638(1-acryloyl-N-(3-(((8-isopropyl-2-((1-methylpiperid...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526639(4-acryloyl-N-(3-(((8-isopropyl-2-((1-methylpiperid...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526640(4-acryloyl-N-(3-(((8-isopropyl-2-((1-methylpiperid...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526641(3-acrylamido-N-(3-(((8-isopropyl-2-((1-methylpiper...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526642((1,4-cis)-4-acrylamido-N-(3-(((8-isopropyl-2-((1-m...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526643(1-acryloyl-N-(3-(((8-isopropyl-2-((1-methylpiperid...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526644(1-acryloyl-N-(2-fluoro-5-(((8-isopropyl-2-((1-meth...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526646(1-acryloyl-N-(3-(1-((8-isopropyl-2-((1-methylpiper...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526647(2-(1-acryloylpiperidine-3-carboxamido)-5-(((8-isop...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526648(3-(((8-isopropyl-2-((1-methylpiperidin-4-yl)oxy)py...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526649((E)-1-(4-(dimethylamino)but-2-enoyl)-N-(3-(((8-iso...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526650((E)-1-(4-(dimethylamino)but-2-enoyl)-N-(2-fluoro-5...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526651((1,4-cis)-4-((E)-4-(dimethylamino)but-2-enamido)-N...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526652(4-acrylamido-N-(3-((8-isopropyl-2-((1-methylpiperi...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526654(1-acryloyl-N-(3-((8-isopropyl-2-((1-methylpiperidi...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526655(N-(1-acryloylpiperidin-4-yl)-3-((8-isopropyl-2-((1...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526656(N-(1-acryloylpiperidin-3-yl)-3-((8-isopropyl-2-((1...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526657((E)-4-(4-(dimethylamino)but-2-enamido)-N-(3-((8-is...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526659((1,4-Trans)-4-((E)-4-(dimethylamino)but-2-enamido)...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526660((E)-N-(1-(4-(dimethylamino)but-2-enoyl)piperidin-3...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526661((E)-N-(1-(4-(dimethylamino)but-2-enoyl)piperidin-4...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526662((1,4-cis)-4-(((E)-4-(dimethylamino)-4-oxobut-2-en-...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526664((E)-4-(dimethylamino)-1-(4-(2-(((8-isopropyl-2-((t...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526666(1-acryloyl-N-(3-(((3-isopropyl-5-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526570(4-acryloyl-N-(5-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526570(4-acryloyl-N-(5-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526570(4-acryloyl-N-(5-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526578(2-acrylamido-N-(3-(((8-isopropyl-2-((tetrahydro-2H...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526532(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526533(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526534(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526534(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526534(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526538(1-acryloyl-N-(3-(((8-isopropyl-2-((1-methylpiperid...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526544(1-acryloyl-N-(3-(((2-(((3S,4S)-3-fluoropiperidin-4...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526545(1-acryloyl-N-(3-(((2-((3-aminocyclohexyl)amino)-8-...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526546(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526548(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526549((R)-1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526550((S)-1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526551(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526552(3-acrylamido-N-(3-(((8-isopropyl-2-((tetrahydro-2H...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526553(4-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526554(4-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526555(N-(3-(((8-isopropyl-2-((tetrahydro-2H-pyran-4-yl)a...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526557(1-acryloyl-N-(3-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526558(1-acryloyl-N-(5-(((8-isopropyl-2-((tetrahydro-2H-p...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Aurigene Discovery Technologies

US Patent
LigandPNGBDBM526559(1-acryloyl-N-(4-fluoro-3-(((8-isopropyl-2-((tetrah...)
Affinity DataIC50: <300nMAssay Description:The ability of compounds to inhibit CDK7 kinase activity was tested in a TR-FRET assay using 5 nM of CDK7/CycH/MNAT1 obtained from Invitrogen, USA. T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 141 total ) | Next | Last >>
Jump to: