Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 5900
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99467(US8497274, 3)
Affinity DataIC50: <300nMAssay Description:MEK phosphorylation inhibition activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99468(US8497274, 22)
Affinity DataIC50: <300nMAssay Description:MEK phosphorylation inhibition activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99472(US8497274, 54)
Affinity DataIC50: <300nMAssay Description:MEK phosphorylation inhibition activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99470(US8497274, 49)
Affinity DataIC50: <300nMAssay Description:MEK phosphorylation inhibition activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99471(US8497274, 32)
Affinity DataIC50: <300nMAssay Description:MEK phosphorylation inhibition activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity mitogen-activated protein kinase kinase 1(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM99469(US8497274, 53)
Affinity DataIC50: <300nMAssay Description:MEK phosphorylation inhibition activity.More data for this Ligand-Target Pair
In DepthDetails US Patent