Compile Data Set for Download or QSAR
maximum 50k data
Found 61 Enz. Inhib. hit(s) with all data for entry = 5978
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38224(US8546380, 1043 | US8633188, 1043)
Affinity DataIC50:  27nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38226(US8546380, 1199 | US8633188, 1199)
Affinity DataIC50:  32nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38220(US8546380, 1100 | US8633188, 1100)
Affinity DataIC50:  37nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103377(US8546380, 165 | US8633188, 165)
Affinity DataIC50:  39.4nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38216(US8546380, 739 | US8633188, 739)
Affinity DataIC50:  49nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38229(US8546380, 127 | US8633188, 127)
Affinity DataIC50:  54nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34552(US8546380, 793 | US8633188, 793)
Affinity DataIC50:  61nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM36793(US8546380, 1244 | US8546380, 1312)
Affinity DataIC50:  130nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103429(US8546380, 1262 | US8633188, 1262)
Affinity DataIC50:  140nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103392(US8546380, 570 | US8633188, 570)
Affinity DataIC50:  149nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103404(US8546380, 786 | US8633188, 786)
Affinity DataIC50:  156nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38222(US8546380, 436 | US8633188, 436)
Affinity DataIC50:  160nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38213(US8546380, 96 | US8633188, 96)
Affinity DataIC50:  163nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34549(US8546380, 1014 | US8633188, 1014)
Affinity DataIC50:  165nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38211(US8546380, 698 | US8633188, 698)
Affinity DataIC50:  165nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38232(US8546380, 1035 | US8633188, 1035)
Affinity DataIC50:  174nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM36406(US8546380, 912 | US8633188, 912)
Affinity DataIC50:  175nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM36407(US8546380, 212 | US8633188, 212)
Affinity DataIC50:  220nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38218(US8546380, 832 | US8633188, 832)
Affinity DataIC50:  222nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM36405(US8546380, 284 | US8633188, 284)
Affinity DataIC50:  229nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38215(US8546380, 822 | US8633188, 822)
Affinity DataIC50:  243nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34551(US8546380, 964 | US8633188, 964)
Affinity DataIC50:  264nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103387(US8546380, 731 | US8633188, 731)
Affinity DataIC50:  278nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38228(US8546380, 73 | US8633188, 73)
Affinity DataIC50:  435nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103413(US8546380, 972 | US8633188, 972)
Affinity DataIC50:  450nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38221(US8546380, 740 | US8633188, 740)
Affinity DataIC50:  505nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103422(US8546380, 1160 | US8633188, 1160)
Affinity DataIC50:  720nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103410(US8546380, 897 | US8633188, 897)
Affinity DataIC50:  816nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38230(US8546380, 309 | US8633188, 309)
Affinity DataIC50:  833nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM35082(US8546380, 1197 | US8633188, 1197)
Affinity DataIC50:  912nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34558(US8546380, 498 | US8633188, 498)
Affinity DataIC50:  930nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34553(US8546380, 625 | US8633188, 625)
Affinity DataIC50:  1.29E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM36326(US8546380, 176 | US8633188, 176)
Affinity DataIC50:  1.48E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34542(US8546380, 220 | US8633188, 220)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM35086(US8546380, 395 | US8633188, 395)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34542(US8546380, 220 | US8633188, 220)
Affinity DataIC50:  1.50E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34559(US8546380, 26 | US8633188, 26)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM36451(US8546380, 163 | US8633188, 163)
Affinity DataIC50:  2.28E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38231(US8546380, 1135 | US8633188, 1135)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103391(US8546380, 504 | US8633188, 504)
Affinity DataIC50:  2.50E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103420(US8546380, 1132 | US8633188, 1132)
Affinity DataIC50:  2.56E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103416(US8546380, 1010 | US8633188, 1010)
Affinity DataIC50:  2.80E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103381(US8546380, 246 | US8633188, 246)
Affinity DataIC50:  2.90E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM34560(US8546380, 465 | US8633188, 465)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM35652(US8546380, 664 | US8633188, 664)
Affinity DataIC50:  3.64E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103427(US8546380, 1207 | US8633188, 1207)
Affinity DataIC50:  4.00E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103414(US8546380, 998 | US8633188, 998)
Affinity DataIC50:  4.50E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM35282(US8546380, 660 | US8633188, 660)
Affinity DataIC50:  4.59E+3nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103386(US8546380, 417 | US8633188, 417)
Affinity DataIC50:  5.00E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103389(US8546380, 490 | US8633188, 490)
Affinity DataIC50:  5.10E+3nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
Displayed 1 to 50 (of 61 total ) | Next | Last >>
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