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Found 5 Enz. Inhib. hit(s) with all data for entry = 7712
TargetBeta-lactamase(Pseudomonas aeruginosa (PAO1))
Meiji Seika Pharma

US Patent
LigandPNGBDBM212440(US8772490, H)
Affinity DataIC50:  650nMpH: 7.0 T: 2°CAssay Description:For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa (PAO1))
Meiji Seika Pharma

US Patent
LigandPNGBDBM159600(US8772490, Example 23 | US9035062, 23)
Affinity DataIC50:  650nMpH: 7.0 T: 2°CAssay Description:For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa (PAO1))
Meiji Seika Pharma

US Patent
LigandPNGBDBM212441(US8772490, TAZ)
Affinity DataIC50:  950nMpH: 7.0 T: 2°CAssay Description:For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa (PAO1))
Meiji Seika Pharma

US Patent
LigandPNGBDBM159601(US8772490, Example 24 | US9035062, 24)
Affinity DataIC50: >3.00E+4nMpH: 7.0 T: 2°CAssay Description:For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-lactamase(Pseudomonas aeruginosa (PAO1))
Meiji Seika Pharma

US Patent
LigandPNGBDBM159601(US8772490, Example 24 | US9035062, 24)
Affinity DataIC50: >3.00E+4nMpH: 7.0 T: 2°CAssay Description:For the measurement of β-lactamase inhibitory activity, 100 uM (final concentration) nitrocefin (Oxoid) was used as a substrate, and 2.5% DMSO, ...More data for this Ligand-Target Pair
In DepthDetails US Patent