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Found 36 Enz. Inhib. hit(s) with all data for entry = 6842
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  5.20nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  6.70nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  27nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153655(US8999994, 7)
Affinity DataIC50:  260nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359397(CHEMBL1929419 | US8999994, 4)
Affinity DataIC50:  310nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153654(US8999994, 6)
Affinity DataIC50:  350nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359396(CHEMBL1929420 | US8999994, 5)
Affinity DataIC50:  420nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153654(US8999994, 6)
Affinity DataIC50:  460nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359394(CHEMBL1929423 | US8999994, 1)
Affinity DataIC50:  800nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153655(US8999994, 7)
Affinity DataIC50:  990nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359397(CHEMBL1929419 | US8999994, 4)
Affinity DataIC50:  1.10E+3nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359396(CHEMBL1929420 | US8999994, 5)
Affinity DataIC50:  2.10E+3nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359393(CHEMBL1926712 | US8999994, 2)
Affinity DataIC50:  2.20E+3nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153654(US8999994, 6)
Affinity DataIC50:  5.20E+3nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359396(CHEMBL1929420 | US8999994, 5)
Affinity DataIC50:  6.70E+3nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  7.40E+3nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359392(CHEMBL1929424 | US8999994, 3)
Affinity DataIC50:  7.60E+3nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153655(US8999994, 7)
Affinity DataIC50:  1.05E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359393(CHEMBL1926712 | US8999994, 2)
Affinity DataIC50:  1.81E+4nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359392(CHEMBL1929424 | US8999994, 3)
Affinity DataIC50:  3.05E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  4.03E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153654(US8999994, 6)
Affinity DataIC50:  4.31E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359393(CHEMBL1926712 | US8999994, 2)
Affinity DataIC50:  6.54E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359397(CHEMBL1929419 | US8999994, 4)
Affinity DataIC50:  8.22E+4nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359392(CHEMBL1929424 | US8999994, 3)
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359394(CHEMBL1929423 | US8999994, 1)
Affinity DataIC50: >1.00E+5nMpH: 8.0Assay Description:The inhibitory activity of the enzyme acetylcholinesterase (AChE) was evaluated by the Ellman method (Biochem. Pharmacol. 1961, 7, 88) using an elect...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359396(CHEMBL1929420 | US8999994, 5)
Affinity DataIC50:  1.30E+5nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359394(CHEMBL1929423 | US8999994, 1)
Affinity DataIC50:  1.43E+5nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8961(1,2,3,4-tetrahydro-9-acridinamine | 1,2,3,4-tetrah...)
Affinity DataIC50:  5.00E+5nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359397(CHEMBL1929419 | US8999994, 4)
Affinity DataIC50:  7.45E+5nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359394(CHEMBL1929423 | US8999994, 1)
Affinity DataIC50:  1.46E+6nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359392(CHEMBL1929424 | US8999994, 3)
Affinity DataIC50:  1.64E+6nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM153655(US8999994, 7)
Affinity DataIC50:  2.77E+6nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM50359393(CHEMBL1926712 | US8999994, 2)
Affinity DataIC50:  1.13E+7nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] B(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  1.54E+7nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Consejo Superior De Investigaciones Cientificas

US Patent
LigandPNGBDBM8960((+/-)-2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimet...)
Affinity DataIC50:  8.55E+8nMpH: 7.4 T: 2°CAssay Description:The inhibitory activity of monoamine oxidases A and B was assessed by the Fowler and Tipton radiometric method (Biochem Pharmacol 1981, 30, 3329) usi...More data for this Ligand-Target Pair
In DepthDetails US Patent