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Found 37 Enz. Inhib. hit(s) with all data for entry = 7138
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177718(US9120780, 24)
Affinity DataIC50:  80nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177712(US9120780, 18)
Affinity DataIC50:  90nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177719(US9120780, 25)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177700(US9120780, 6)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177702(US9120780, 8)
Affinity DataIC50:  110nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177746(US9120780, 49)
Affinity DataIC50:  120nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177706(US9120780, 12)
Affinity DataIC50:  120nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177714(US9120780, 20)
Affinity DataIC50:  140nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177716(US9120780, 22)
Affinity DataIC50:  140nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177715(US9120780, 21)
Affinity DataIC50:  150nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177748(US9120780, 51)
Affinity DataIC50:  160nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177698(US9120780, 4)
Affinity DataIC50:  160nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177695(US9120780, 1)
Affinity DataIC50:  170nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177713(US9120780, 19)
Affinity DataIC50:  170nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177743(US9120780, 46)
Affinity DataIC50:  190nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177707(US9120780, 13)
Affinity DataIC50:  200nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177709(US9120780, 15)
Affinity DataIC50:  230nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177699(US9120780, 5)
Affinity DataIC50:  240nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177704(US9120780, 10)
Affinity DataIC50:  250nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177747(US9120780, 50)
Affinity DataIC50:  250nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177745(US9120780, 48)
Affinity DataIC50:  260nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177703(US9120780, 9)
Affinity DataIC50:  260nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177708(US9120780, 14)
Affinity DataIC50:  270nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177717(US9120780, 23)
Affinity DataIC50:  280nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177710(US9120780, 16)
Affinity DataIC50:  290nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177705(US9120780, 11)
Affinity DataIC50:  300nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177701(US9120780, 7)
Affinity DataIC50:  370nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177749(US9120780, 52)
Affinity DataIC50:  420nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177744(US9120780, 47)
Affinity DataIC50:  430nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177711(US9120780, 17)
Affinity DataIC50:  490nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177697(US9120780, 3)
Affinity DataIC50:  740nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177750(US9120780, Comparative Example 3)
Affinity DataIC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177751(US9120780, Comparative Example 4)
Affinity DataIC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM126164(US8779142, Comparative Example 1 | US9120780, Comp...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM126165(US8779142, Comparative Example 2 | US9120780, Comp...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM177752(US9120780, Comparative Example 5)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetHeat shock protein HSP 90-alpha(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM126169(US8779142, Comparative Example 6 | US9120780, Comp...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The HSP90-binding activity was measured by an AlphaScreen competitive assay system. The purified HSP90 solution was diluted with a binding buffer (50...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent