Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 7404
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192964(US9193697, B5.2)
Affinity DataIC50:  4.19nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM193011(US9193697, C6.2)
Affinity DataIC50:  8.68nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192971(US9193697, B5.9)
Affinity DataIC50:  9.61nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM193010(US9193697, C6.1)
Affinity DataIC50:  11.9nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192965(US9193697, B5.3)
Affinity DataIC50:  12.8nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192973(US9193697, B5.11)
Affinity DataIC50:  13.1nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM193012(US9193697, C6.3)
Affinity DataIC50:  15.9nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192963(US9193697, B5.1)
Affinity DataIC50:  17.9nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192932(US9193697, A7.21)
Affinity DataIC50:  25.9nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192966(US9193697, B5.4)
Affinity DataIC50:  27.6nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192933(US9193697, A7.22)
Affinity DataIC50:  45.8nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192934(US9193697, A7.23)
Affinity DataIC50:  61.7nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192925(US9193697, A7.14)
Affinity DataIC50:  65.3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192924(US9193697, A7.13)
Affinity DataIC50:  67.5nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192972(US9193697, B5.10)
Affinity DataIC50:  67.6nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192928(US9193697, A7.17)
Affinity DataIC50:  75.1nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192969(US9193697, B5.7)
Affinity DataIC50:  92.2nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192974(US9193697, B5.12)
Affinity DataIC50:  113nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192968(US9193697, B5.6)
Affinity DataIC50:  118nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192970(US9193697, B5.8)
Affinity DataIC50:  146nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192935(US9193697, A7.24)
Affinity DataIC50:  201nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192967(US9193697, B5.5)
Affinity DataIC50:  255nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192930(US9193697, A7.19)
Affinity DataIC50:  287nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192913(US9193697, A7.2)
Affinity DataIC50:  293nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192975(US9193697, B5.13)
Affinity DataIC50:  320nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192938(US9193697, A7.27)
Affinity DataIC50:  482nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192936(US9193697, A7.25)
Affinity DataIC50:  525nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192937(US9193697, A7.26)
Affinity DataIC50:  748nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192929(US9193697, A7.18)
Affinity DataIC50:  839nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192927(US9193697, A7.16)
Affinity DataIC50:  925nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192926(US9193697, A7.15)
Affinity DataIC50:  1.42E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192931(US9193697, A7.20)
Affinity DataIC50:  1.70E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192940(US9193697, A7.29)
Affinity DataIC50:  1.91E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192941(US9193697, A7.30)
Affinity DataIC50:  2.14E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192942(US9193697, A7.31 and A7.31a)
Affinity DataIC50:  2.22E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192939(US9193697, A7.28)
Affinity DataIC50:  3.09E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192977(US9193697, B5.15)
Affinity DataIC50:  4.53E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192976(US9193697, B5.14)
Affinity DataIC50:  9.15E+3nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM192942(US9193697, A7.31 and A7.31a)
Affinity DataIC50:  1.00E+4nMAssay Description:Enzyme activity was demonstrated in a radioenzymatic test based on measuring the product of hydrolysis (ethanolamine [3]H) of anandamide [ethanolam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent