TargetcGMP-specific 3',5'-cyclic phosphodiesterase [535-860](Homo sapiens (Human))
University Of North Carolina At Chapel Hill
University Of North Carolina At Chapel Hill
Affinity DataIC50: 2.10E+3nMpH: 7.8 T: 2°CAssay Description:Enzymatic activity of the isolated catalytic domains of wild type PDE5A1 and its deletion mutants was assayed by using [3H]cGMP as substrate in a rea...More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase [1-662,679-875](Homo sapiens (Human))
University Of North Carolina At Chapel Hill
University Of North Carolina At Chapel Hill
Affinity DataIC50: 5.30E+3nMpH: 7.8 T: 2°CAssay Description:Enzymatic activity of the isolated catalytic domains of wild type PDE5A1 and its deletion mutants was assayed by using [3H]cGMP as substrate in a rea...More data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Institute Of Pharmaceutical Chemistry
Curated by ChEMBL
Institute Of Pharmaceutical Chemistry
Curated by ChEMBL
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of PDE5 from plateletsMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase [1-660,682-875](Homo sapiens (Human))
University Of North Carolina At Chapel Hill
University Of North Carolina At Chapel Hill
Affinity DataIC50: 9.50E+4nMpH: 7.8 T: 2°CAssay Description:Enzymatic activity of the isolated catalytic domains of wild type PDE5A1 and its deletion mutants was assayed by using [3H]cGMP as substrate in a rea...More data for this Ligand-Target Pair