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Found 2 Enz. Inhib. hit(s) for PDB: 1UK1
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM27714(5-fluoro-1-[4-(4-phenyl-1,2,3,6-tetrahydropyridin-...)
Affinity DataIC50:  60nMAssay Description:In vitro inhibitory concentration against human recombinant Poly (ADP-ribose) polymerase 1More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Fujisawa Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM27714(5-fluoro-1-[4-(4-phenyl-1,2,3,6-tetrahydropyridin-...)
Affinity DataIC50:  60nMpH: 8.0 T: 2°CAssay Description:To assess the inhibitory activity of novel inhibitors, the PARP enzyme assay was carried out in reaction mixture consisting of activated salmon teste...More data for this Ligand-Target Pair