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Found 2 Enz. Inhib. hit(s) for PDB: 2BYQ
TargetSoluble acetylcholine receptor(Aplysia Californica)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50049757(()-2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]h...)
Affinity DataKi:  1nMAssay Description:Binding affinity to salt water mollusc Aplysia californica AChBP Y55W mutant assessed as [3H]acetamiprid binding by radioligand binding assayMore data for this Ligand-Target Pair
TargetSoluble acetylcholine receptor(Aplysia Californica)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50143314((+)-Epibatidine | (-)-epibatidine | (1R,2R,4S)-2-(...)
Affinity DataKi:  7.40nM ΔG°:  -45.6kJ/molepH: 7.4 T: 2°CAssay Description:Assay Description 2 Assays used to generate Ki or EC50 values. 1) SPA Assay - Quick screen binding assays were performed using 100 ul of 0.2 mg/ml an...More data for this Ligand-Target Pair
In DepthDetails PDB3D3D Structure (crystal)