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Found 1 Enz. Inhib. hit(s) for PDB: 2CGV
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
Vernalis (R&D)

LigandPNGBDBM14821((2S)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan...)
Affinity DataIC50:  2.73E+4nMpH: 7.5 T: 2°CAssay Description:Chk1 kinase activity was assayed in reaction buffer containing substrate peptide, enzyme, and inhibitor in the presence of 100uM ATP/[gamma-33P] ATP....More data for this Ligand-Target Pair