TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataIC50: 0.690nMAssay Description:Inhibition of ASK1 (unknown origin) by HTRF assayMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding constant for MAP3K5 kinase domainMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataKd: 120nMAssay Description:Average Binding Constant for MAP3K5; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Zhejiang University
Curated by ChEMBL
Zhejiang University
Curated by ChEMBL
Affinity DataKd: 110nMAssay Description:Binding constant for ASK1 kinase domainMore data for this Ligand-Target Pair